c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cn1c(Cl)cc2ccc(Nc3cccc(-n4cncn4)c3)nc21
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cn1ncc(Nc2ccccc2Cl)c1-n1nnc2ccccc21
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC CCCc1nn(-c2nc3[nH]c(C)c(C)n3n2)c2ccc(Cl)cc12
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC CCc1cc(Cl)nc(-c2n[nH]c3ccc(-n4cncn4)cc23)c1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC CC=C(C)Cn1c(Cl)cc2c3c(ncc31)[nH]c1c(C#N)cnn12
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC CCc1cnn(Cc2c[nH]c(-n3ncc4ccccc43)n2)c1Cl
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC CCCn1nc(C)c2nc3[nH]c4nc(CCCCl)cn4c3cc21
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cc1cccc(-n2cc(Nc3nnc4ccc(Cl)cn34)cn2)c1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Clc1cnccc1Nc1ccc2nc(-n3cncn3)ccc2c1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cc1cc2cnn3c(Nc4cncc(Cl)c4)nnc3c2cc1C
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cn1c(NN=Cc2ccc3[nH]ccc3c2)nc2cnc(Cl)cc21
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cc1nn(-c2nccc(-c3cc(C)c4cc[nH]c4n3)n2)cc1Cl
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cc1cn2cc(Nc3nncn3-c3cccnc3)ccc2c1Cl
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC C=CC(=CC)Nc1n[nH]c2nc3nc4cc(Cl)ccc4n3cc12
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cc1ccc(C(Cl)=CCc2nc3c(ccn4nnnc34)[nH]2)cc1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC ClCc1cccc(-n2ccc(Nc3cnc4ccncn34)n2)c1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC CCc1cc(CNc2nnc3c4cccn4ccn23)cc(Cl)n1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cc1cn(-c2ccc3nc(C)cc(-n4cccn4)c3c2Cl)nn1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Clc1cc(-n2cnnc2-c2ccc(-c3cn[nH]c3)cc2)ccn1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC CCC=Nc1nc2[nH]cnc2c2cc(-c3ccc(Cl)cc3)nn12
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Clc1ccc(-c2cc(-c3ccc(-n4cccn4)nn3)n[nH]2)cc1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Clc1[nH]cnc1CNc1cccc(-c2ccn3cnnc3c2)c1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC CCn1c(-c2ccccc2)nn2c(Cc3[nH]ccc3Cl)nnc12
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Clc1cn(-c2c[nH]c(-c3ncccc3-n3cccc3)n2)cn1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cn1cc(Nc2cc3ccc4cnc(Cl)cc4n3n2)ccc1=N
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC C=Nc1nn(-c2n[nH]c(-c3ccccc3Cl)n2)c2ccccc12
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cc1nc2cccc(Cl)c2c2nnc(CNc3cccnc3)n12
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cc1[nH]nc2c1[nH]c1cc(N(C)Cc3cccc(Cl)c3)nn12
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC Cc1cn2cccc(-c3n[nH]c(C(Cl)c4ccccn4)n3)c2n1
c12n(nc(n1)c1c(Cl)cccc1)c(nc1c2nc[nH]1)CCCC CCN(C)c1ccc(-c2nn3c(nc4cc(Cl)ccc43)[nH]2)nc1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cc1ncnc2c1ccn2Cc1ccc2c(n1)[nH]c1ccccc12
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 C(=Cc1ccc2cn[nH]c2n1)CCc1nc2cccc3ccn1c32
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cc1cc(C=c2cc3c4ccccc4nc3n3ccnc23)cnn1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cc1cc2c3c(nncc3c(C)n2-c2ccnc3ccccc23)[nH]1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 CC=C(C)C=Cc1cc2c3ccn4cc5ccnc(n2n1)n5c34
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 C=C1Cc2cc3c(nc2C1=CC)c(-n1cccn1)nc1nccn13
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 c1ccc2c(Nc3nnc4c5ccccc5cnn34)cccc2c1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 CC=c1cncnn(C)c2nc3ccccc3n2c2ccc1cc2
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 C1=Cc2nc(C=Cc3cnc4c(cnc5nccn54)c3)ccc2C1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cn1ccnc1Cn1c2ccccc2c2nc3ccccn3c21
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cc1ccc2c(-n3nncc3C)cc(C=Cc3cc[nH]n3)cc2c1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 C=CN(C)c1nc2c(=C)c(=C)ncc2c2nc3cc(C)ccn3c12
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 C=C(C)C=Cc1cc(-c2nnc[nH]2)cc2c1ccc1cnn(C)c12
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cc1cccc2c3cc4c(nc3cn12)c1cnn2c1n4CC(C)C2
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 c1ccc(-c2cnn3c(-c4cc5ccccc5[nH]4)nnc3c2)cc1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 CN=c1c(C)ccc[nH]c2ccc3c(cccc3c3ncnn13)c2
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cc1cc2cc3c(cc2n1Cc1cn2ccccc2n1)ncn3C
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 c1ccc2cc(-c3cn(-c4ccc5[nH]cnc5c4)nn3)ccc2c1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cn1cc(CCc2[nH]c3ccccc3c2C=Nn2cccc2)cn1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 C=CC(=C)C=Cc1cccc(-n2ncc3cn4ccnc4cc32)n1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 C(=Nc1ccc2c(ccn3c4ccccc4nc23)n1)C1=NCCC1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 CC=CC=c1c(=Nc2cnn(C)c2)c2ccccc2n2ccnc12
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 N#Cc1cccc(C(N=Cc2cn[nH]c2)=c2ccn3cccc23)c1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 c1ccc2c(c1)cc(-c1nc3ccccc3[nH]1)n2Cc1cn[nH]c1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cc1cc2ncnn2c2nc(C#N)c3cc4ccccc4cc3c12
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 CNC(=O)C=Cc1cnc2c3cccc(-n4cccn4)c3ccn12
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 C=CCn1c2ccccc2c2ccc(-n3nnc(=C)c3=CC)nc21
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Cn1ccc(-c2nc3nc4ccccc4cc3c3nn(C)cc23)c1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 Nc1ccc2ccc(-c3nnc4c5ccccc5cnn34)cc2c1
n12c(nc(n1)c1ccccc1)c1c(nc2c2ccccc2)nc[n-]1 c1ccc2c(-c3ccc(-c4nc5[nH]ncn5n4)cc3)cccc2c1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 CC=C(S)CNc1ccc2c(n1)c(=O)nc1sc3ccccc3n12
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 O=[SH]c1ccc(C=NNc2ncc3c(ccc4ccccc43)n2)s1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cc1ccc(-n2c(SCc3nc4ccccc4s3)n[nH]c2=O)cc1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cc1cc(Nc2nccc3cc4cnc(C)n4cc23)sc1C[SH]=O
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cn1c(=NC(=O)CSc2nc3ccccc3[nH]2)sc2ccccc21
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 CCSc1nc2scc(-c3ccc(C)c4ccnnc34)c2c(=O)[nH]1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 CSc1nccc2c(C(=O)N=c3sccn3C)cc3cc[nH]c3c12
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 O=C(N=c1[nH]c2ccccc2s1)c1cnn(-c2cccc(S)c2)c1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 CCSCc1cc2c(s1)c(=O)[nH]c1nc(-c3cccnn3)ccc12
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 O=C(CSCc1nc2sc3ccccc3n2n1)Nc1ccccc1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 O=c1ccc(Nc2ccc(-c3csc4ccccc34)cn2)nn1S
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cn1ccc(-c2ccc3nc(-c4ccc(N[SH]=O)cc4)sc3c2)n1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 CSc1nc2ncc(C(=O)Nc3ccc4ccccc4c3)nc2s1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 COc1ccc(-c2csc3ncnc(SCc4ncc[nH]4)c23)cc1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cc1ccc2sc(=NC(=O)c3sc(C)c4c3ncn4C)[nH]c2c1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 CS(=O)Nc1ccc2cnn(-c3ccc(-c4ccns4)cc3)c2c1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cc1csc(Nc2nnc(COc3cccc4ccccc34)s2)n1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Oc1ccc(Sc2nnc(-n3ccnc3-c3ccccc3)s2)cc1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 CCn1c2ccc(S)cc2c2cc(C(=O)Nc3nncs3)ccc21
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cc1ccnn1-c1cccc2c(=S)nc(SCc3ccco3)[nH]c12
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 C=NC(=CC)c1nc(C(=O)N=c2sc3cccc4ccn2c43)cs1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cn1c(SC(c2cn[nH]c2)c2cccs2)nc2ccccc2c1=O
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 O=c1[nH]nc2scc(-c3ccc(N=Cc4ccc(S)cc4)cc3)n12
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 c1csc(COc2ccc3ccc(CSc4nnn[nH]4)cc3c2)c1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cc1ccccc1CSCc1nc2[nH]c3cc([SH]=O)ccc3n2n1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 Cc1n[nH]c(SCc2nc(-c3c(C)oc4ccccc34)cs2)n1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 O=S(Cc1cccc2sc(=Nc3ccccc3)[nH]c12)c1cn[nH]c1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 COc1cc(C)ccc1-c1n[nH]c(-n2c(=S)sc3ccccc32)n1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 SCc1cn(-c2ccc3nc4sc5c(c4cc3c2)COCC5)nn1
n1c(nc(c2c1ccs2)C(=O)c1sccc1)NCc1cccnc1 C=S(C)(=O)Nc1ncc2sc(-c3cccc4ccccc34)nc2n1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 c1ccc2oc(CSc3nnnn3-c3ccsc3)nc2c1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Sc1nncn1-c1nc(Cc2csc3ccccc23)no1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Cc1ccc(Sc2nnnn2-c2csc3cnoc23)cc1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Cc1cc2c(ccc(=O)n2-c2nnc(-n3cccn3)s2)s1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 c1ccn2cc(-c3nc(CSc4cocn4)ns3)nc2c1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 COc1ccc2sc(-c3nc(-n4cncn4)ns3)cc2c1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 N#CCSc1nc(=O)n2ccc3[nH]c4sccc4c3c2n1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 c1ccc2oc(Cc3nnc(Nc4nncs4)s3)cc2c1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 c1ccc2oc(CSCc3nn4cnnc4s3)cc2c1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Cc1nnc(-c2ccccc2Sc2nnc3sccn23)o1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Oc1cncc(CSc2nnc3sc4ccccc4n23)n1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 CSc1nn(C)cc1-c1nnc2sc3ccc(O)cc3n12
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 CSc1nnc(-c2csc(-n3cnc4ccccc43)n2)o1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Cc1csc(-n2nnnc2-c2csc(-c3cnoc3)c2)c1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Cc1nocc1CCSc1nnc2c3scnc3ccn12
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Oc1ccnc2ccc(SCc3csc4nnnn34)cc12
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Cc1nn(-c2nc3c(cnn3-c3ccccc3)s2)c(=O)s1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 CC(SCc1cc2nnn3ccoc(n1)c23)c1cscn1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Cc1cn2c(C(C)Sc3ccc4ncoc4n3)nnc2s1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Oc1ccc2nc(Nc3nnc(-n4cccc4)s3)sc2c1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 COc1cccc(-c2nc3nn4c(S)nnc4cc3s2)c1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Cc1ccn2c(Sc3nnc(-c4ccco4)s3)nnc2c1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 Cc1nc2nc(CSc3nc4n(n3)COC=C4)ccc2s1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 CC1OCC=Cn2nc(Sc3ncnc4sccc34)nc21
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 CC(Sc1nnc2n1-c1ccccc1OC2)c1nncs1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 N#CCc1ccc(C=C2c3sccc3Sc3nnnn32)o1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 CC=Cn1nnnc1Sn1c(=O)c(S)cc2ccccc21
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 C=CC1=CCC(=O)N1c1nnc(-n2ncc3ccsc32)s1
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 O=c1c(=Cc2cn3ccsc3n2)sc2nnc(C3CC3)n12
c1nc2c(sc(=S)n2CC=C)c2n1nc(n2)c1occc1 CCS(=O)n1ccc2nc(-c3cn4cnnc4s3)ccc21
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N N#CCNC(=O)Nc1cc2ccccc2c2ccccc12
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N O=c1ccc2nc3cc(C4=CNCC=C4)ccc3cc2[nH]1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N N#Cc1cc(C(=O)NCc2cccc3ccccc23)c[nH]1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N O=c1[nH]c2ncccc2c2ccc(NCC3=CCC3)cc12
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N N#Cc1cccc(CNC(=O)c2cc3ccccc3[nH]2)c1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N C(=Cc1nc2ccccc2[nH]1)c1ccc2c(c1)CNCO2
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N O=C(Nc1ccc2c3c([nH]c2c1)CCC3)c1ccncc1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N O=C(Nc1ccc2cc[nH]c2c1)c1ccc2c(c1)CNC2
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N CC1=C(C)Cc2c([nH]c(=O)c3c2[nH]c2cccnc23)CC1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N Cc1cccc(C=NNC(=O)c2ccc3cc[nH]c3c2)c1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N O=C(Nc1cnc2c(c1)=CCC=2)c1cc2ccccc2[nH]1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N C=CC=NC(=O)c1c[nH]c2ccc(-c3ccc(C)[nH]3)cc12
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N C=C(C)C=CNc1ccc2c(=O)[nH]c3ccncc3c2c1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N C#CCc1ccc(C(=O)N=c2[nH]c3ccccc3[nH]2)cc1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N Nc1c2c(cc3cccc(-n4cnc(C=O)c4)c13)CCC2
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N N#Cc1c(NCc2ccccc2)[nH]c(=O)c2ccccc12
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N Cc1[nH]ccc1C(=O)Nc1ccc(C#N)c2ccccc12
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N CCC1Cc2ccc(-c3nc4[nH]c(=O)ccc4[nH]3)cc2C1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N O=c1[nH]c2c(c3[nH]nc(-c4ccccc4)c13)CC=CCC2
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N Cc1ccccc1C=NNC(=O)c1cc2ccccc2[nH]1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N Cc1cc(C)c2oc(C=C3NCc4ccnnc43)cc2c1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N N#CC(=Cc1cccc2cc[nH]c12)c1cc(O)ccn1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N Nc1ccn(-c2ccc(-c3ccc4c(c3)CCO4)cc2)n1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N c1ccc(-c2n[nH]cc2-c2ccc3c(c2)NCCO3)cc1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N C=CC(=CC)NCc1ccc2[nH]c3c(=O)[nH]ccc3c2c1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N c1ccc2c3c(cc(NCc4cocn4)c2c1)CNCC3
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N c1ccc2c(Nc3ccc4c(c3)NCCO4)ccnc2c1
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N O=c1nc(Nc2ccc(C3CC3)cc2)[nH]c2ccccc12
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N O=C1Nc2ccccc2Nc2ccc(-n3cccc3)cc21
c12c(c3c(C1=O)cccc3)nc(nc2c1ccccc1)N C=CCNC(=O)c1c[nH]nc1-c1cccc2ccccc12
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N C=C(N)C1COc2cc3ccc4cn[nH]c4c3cc2O1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N CNC(=O)Nc1ccc2[nH]c(=O)c3ccccc3c2c1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N COc1ccc(N=c2[nH]c(=O)c3ccccc3[nH]2)cc1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N Nc1c2ccccc2cc2nc(N3CCOCC3)oc12
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N Cc1cc2c(cn1)CC(c1cccc3oc(=O)[nH]c13)N2
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N CC(=O)Nc1cccc(-n2c(=O)[nH]c3ccccc32)c1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=c1[nH]c(C=Nc2ccccc2)nc2c(O)cccc12
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=C(Cn1ccccc1=O)Nc1cccc2[nH]ccc12
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=C1N=C(Nc2ccc3oc4ccccc4c3c2)CN1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=C(Nc1nc2ccccc2[nH]1)c1cc2c(o1)CCC2
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=c1cc(C2=CCOC=C2)n2nc3ccccc3c2[nH]1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=C(Nc1ccccc1)c1ccc2c(=O)[nH]ncc2c1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N CC1Cc2cc3ccc4[nH]c(N)nc(=O)c4c3cc2O1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N C=CCOc1ccc2c(c1)[nH]c(=O)c1c(CC)[nH]nc12
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N CN=c1[nH]ccc2ccc(NC(=O)c3ccco3)cc12
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N Oc1ccc(-c2nnc3cc4c(cn23)CCC4)cc1O
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N CNc1cccc(C(=O)n2[nH]c(=O)c3ccccc32)c1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=C(Nc1cccc2cc[nH]c(=O)c12)c1ccncc1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=c1[nH]c(C(O)C2CC2)nc2ncc3ccccc3c12
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=C(C=Cc1c[nH]c2cc(=O)[nH]nc12)c1ccccc1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=Cc1ccc(C(=O)Nc2ccc3[nH]cnc3c2)cc1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N Nc1ccc(Oc2ccc3oc4c(c3c2)C=CC4)nn1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N Cc1nc(C=CC(=O)Nc2cccc3[nH]ccc23)co1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=C(Nc1ccc[nH]c1=O)c1cccc2cnccc12
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N C=CCNc1ccc2nc(-c3ccc[nH]c3=O)oc2c1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N c1cc(-c2ccc(-c3ccc4c(c3)OCCN4)o2)n[nH]1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N O=C(Nc1ccc2c(=O)[nH]ccc2c1)c1cccnc1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N CCNC(=O)c1cc2c(=O)c3cc(C)ccc3[nH]c2[nH]1
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N CC=C(C)c1nc(=O)c2ccccc2c2cc(=O)[nH]n12
c1ccc2c(c1)C(=O)c1c2nc(nc1c1occc1)N Cc1nc(COC(=O)c2cc3ccccc3[nH]2)[nH]c1C
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1cc(-c2cc3cncc(-c4nc5c(C)nn(C)c5[nH]4)n3n2)ccc1O
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1nn(C)c(Nc2cnc3nn[nH]c3c2)c1Cc1coc2ccccc12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 O=c1cc(N(Cc2c[nH]nn2)c2ccc3ccccc3c2)nc2[nH]ccn12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CC(Nc1cnc2[nH]c(=O)c3ccccc3n12)c1ccc2c(ncn2C)n1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cn1nccc1CNc1cc2c(cn1)[nH]c1nc3ccc(O)cc3nc12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1n[nH]c2nc3cnccc3c(COc3ccc(-c4nc[nH]n4)cc3)c12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1cc2nnc(C(=O)NCc3ccc4ccccc4c3)c3nnc([nH]1)n23
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 OCc1nc2ccc(C=Nn3c(-c4cn[nH]c4)nc4ccccc43)cc2[nH]1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CCc1ccc(Nc2ncn3c2c(=O)[nH]c2nccnc23)c2cccnc12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CCNc1nc2n(n1)c(=Nc1ccc(C)cc1)c1cccc3[nH]c(=O)n2c31
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CNc1nc(=O)c2nn(-c3ccc4ccc5ccccc5c4c3)nc2[nH]1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CCc1nc(-c2cnc3nc4ccccc4n3c2-c2ccnc(N)c2)no1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cn1nnn2ccc(-c3ccc(NC(=O)c4ccc5nc[nH]c5c4)cc3)c12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1cccc2[nH]c(=Nc3nc4[nH]nc(-c5ccc(O)cc5)n4n3)ccc12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 c1ccc(-c2nnc(CNc3cc(-c4nn5cccc5[nH]4)ccn3)o2)cc1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CCn1cnc2c3c(cc(N)nc31)nn2-c1ccc(-n2cccc2)cc1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CC=CNc1cc2nc(-c3ccccc3)cn2c2nc3[nH]cnn3c(=O)c12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1nn2c(cc1NC(=O)c1cccn3cnnc13)cc1ccc(N)cc12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1ccc(-n2nc(-c3ccc[nH]3)c3c(=O)n(C)n4ccnc4c32)nc1C
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CCc1nc(-c2cccc(N=c3[nH]c4ccccc4c4cnnn34)c2)no1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 C=NC(=CC)N=c1[nH]c2ccc(OCC)cc2c2nnc(-c3cc[nH]c3)n12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1cnc(NN=Cc2ccc3[nH]c(=Nc4nccn4C)oc3c2)c(C)c1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CCCn1cc(Nc2cc(-c3ccnc4nc5ccccc5n34)on2)cn1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cn1c2ccccc2n2ncc(C(=O)Nc3nnc(-c4ccccc4)[nH]3)c12
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1ccc(NC(=O)c2ccncn2)c(C=Nn2c(C)cc3cc[nH]c32)n1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 OC1CCNC1=NC=Cc1nc2cc3ccc(-n4ccnc4)nc3cc2[nH]1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 CON=Cc1cc2ccc(C)cc2[nH]c1=Nc1cnn(-c2ncc[nH]2)c1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 c1ccc(-c2nc(-c3cn[nH]c3Nc3ccc4cnccc4n3)no2)cc1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1ccc2nc3ncc(N=Cc4cccc(O)c4)c4ncnc(c34)n2n1
n12c(c3c(nc2N)nn(c3)CCCc2ccccc2)nc(n1)c1occc1 Cc1ccn2c(c1)nc1cc(NC(=O)c3nccn4ncnc34)ccc12
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCC(C)n1cc(CN(C)C(=O)c2n[nH]c3ccccc23)c(C(=O)OC)n1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C COc1ccccc1Nc1nnc(CN(C)c2cccc(OCC#N)c2)o1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCCN1C(=O)c2[nH]c3ccc(Oc4nnc(CC)n4CC)cc3c2C1=O
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCC(COC(=O)Cc1cc(C)cc(-n2nnc3cncnc32)c1)=C(C)O
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCCn1cc(C(=O)C=Cc2c[nH]nc2-n2cc(C(=O)OCC)cn2)cn1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCCN(C)c1ncc2ccoc2c1C=C(C#N)OC(=O)Cc1cc[nH]n1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C C=CCN(Cc1cc[nH]c1)C(=O)c1cc(-n2cnc(C)c(CC)c2=O)no1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C COCC(=O)N(C)C=CCNc1nnc(-c2cc(C)nc3ccccc23)o1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C COc1cccc(COc2nnnn2CC(=O)Nc2cc(C)ccc2C)c1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCc1cccc(Oc2ccc(C(=O)Nc3ccn(CCOC)n3)nn2)c1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCOc1cc(-c2cc(C)n[nH]2)ccc1OC(=O)CCCn1ncnc1C
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C COCCOc1ncc(C=CC(=O)Nc2cc(C)cc3cnn(C)c23)cn1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCn1nccc1COc1ccc(OCC(=O)Nc2cnn(C)c2C)cc1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CC(=CC(=O)N=c1[nH]c2ccccc2n1C)n1cc(C=O)nc1OC(C)C
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C Cn1nc(CCC(=O)Nc2ccc(OCC3CC3)cc2)cc1-c1cnno1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CNCC(=Cc1cnc(COc2ccc(C=O)nc2C)o1)c1nccn1C
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C C=CCOCCn1nnc2cc(NC(=O)c3c(C(C)C)noc3C)ccc21
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CC=C(C#N)C(=O)NCCCc1nc(COc2ccc3cc[nH]c3c2)no1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C Cc1noc(CN(CCc2cccn2C)C(=O)NC(C)c2ccco2)n1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCOC(=O)c1cnc(NCC(C)Oc2ccccc2)cc1-n1cncn1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C COc1cccc(NC(=O)Cc2noc(CN(C)c3cc(C)ccn3)n2)c1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CC=C(C)n1ncnc1N=Cc1ccc(OCc2cc(C)n[nH]2)c(OC)c1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C Cc1n[nH]c(C(=O)N(C)CCOc2ccccc2-c2cnc(C3CC3)o2)n1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C COc1nccc2ccc(C(=O)CNC(=O)c3cc(C)n(C(C)C)n3)nc12
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C C=Nn1ccccc1=NOc1cccc2c(C(=O)NC(C)C(C)C)onc12
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C COc1ccc(NC(=O)c2ccn(C)n2)cc1N=Cc1cnc(C(C)C)o1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCOC(=O)c1cc(C)ccc1Nc1nnc(COc2ccncc2)n1C
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCOc1ccc(-n2nnnc2CNC(=O)c2cc(C)ccc2OC)cc1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C CCOc1cc(C)n2ncc(CN(C)C(=O)Nc3ccc(OC)cc3)c2n1
c1(nc(cc(n1)c1cc(cc(c1)OC)OC)NC(=O)C)n1c(cc(n1)C)C Cc1ccccc1OCCOc1cccc(-n2cnc(CCNN=O)n2)c1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 CC=CC=Cc1nnc2n1nc1ccc(C(=O)O)cn12
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 C=CC(=CC)c1n[nH]c(-n2c(=O)ccc3oncc32)n1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 C=Nn1ncc2ccc(OC(=O)c3cc(C)n[nH]3)cc21
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cc1ccc(C=Cc2nncn2-c2cc[nH]c(=O)n2)o1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cn1nccc1C(=O)OCc1ccnn1-c1cc[nH]c1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 C=Nn1c(N=c2cc(C)oc3ccccc23)n[nH]c1=O
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cc1cc(Oc2cc(O)ccn2)nc(-n2cccn2)n1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cn1occ(C=Nc2ccc(-c3ccn[nH]3)cn2)c1=O
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 CCn1ncc2cc(NC(=O)Cc3nnco3)ccc21
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Oc1cc(OCc2nncn2-c2ccccc2)ncn1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 COc1nccn1N=Cc1cc2ccncc2[nH]c1=O
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cc1cc(NC(=O)c2ccc(-n3ccnc3)nc2)on1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cc1occ(O)c1C=Nc1cnnn1-c1ccncc1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 C=CCOC(=O)c1nc2[nH]c(-c3ccncc3)cn2n1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cc1ccc(C(=O)Nc2nnnn2-c2ccccc2)o1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 CCC(=O)n1ccc2c(Oc3cn[nH]c3)nc(C)nc21
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 CCn1cc(-c2nnc(-c3ccc(=O)[nH]c3)o2)c(C)n1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 COc1cc(-c2cc3[nH]ncn3n2)ccc1OCC#N
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cc1cc(C)nc(-n2nc3occ4c3c2CC(=O)N4)n1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cc1ccc(C(=O)N=c2[nH]ncn2-c2ccncc2)o1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cc1ccc(CN(C=O)Cc2cn3c(C)n[nH]c3n2)o1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 COC(=O)c1c[nH]cc1-c1ccc(-n2cccn2)nn1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 CCn1ncc2cc(C(C)=O)c(=O)n(-c3ccn[nH]3)c21
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 O=C(Nc1cccc(Oc2ccccc2)c1)n1nn[nH]1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cn1cnc(COc2nc(=O)[nH]c3ccccc23)c1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cc1ncn2ccnc2c1NC(=O)Oc1cccnc1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 CN=CNc1ncc2c(=Cc3ccc(C=O)o3)cnn12
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 Cn1ccc2cccc(NC(=O)Cn3ccnn3)c21
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 COc1ccccc1Oc1ccc(-n2nnnn2)cc1
o1c(ccc1)c1nc(cc(n1)NC(=O)C)n1nccc1 CN(Cc1c[nH]nn1)C(=O)c1cc2ccccc2o1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Cc1cc2nc(N=C(N)c3nc4ncc(F)cn4c3N)ccc2o1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N CCc1cc(OCCF)c2c(n1)[nH]c1nc(N)nc3[nH]nc2c31
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N COc1ccc(Nc2ncnc3nc(N)c4[nH]ncc4c23)cc1F
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Cc1cc(-c2n[nH]c(=Nc3ccc4[nH]c(=O)[nH]c4n3)[nH]2)ccc1F
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N CC(N)c1ccc(F)cc1C(O)c1n[nH]c2nn3cnnc3cc12
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N O=c1[nH]nc(-c2ccc(-c3cc(CCF)n[nH]3)cc2)c2nn[nH]c12
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Oc1ccc(Cc2cc(-n3ncc(-c4cn[nH]c4)n3)[nH]n2)c(F)c1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N O=C(Nc1cc(CF)n[nH]1)c1c[nH]nc1-c1cccc2c[nH]nc12
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Oc1cc(Nc2nnc(Nc3ccc(F)cc3)[nH]2)c2cc[nH]c2n1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Nc1cnccc1N=c1c2cc(F)ccc2[nH]c2nc(CO)nn12
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N N#Cc1cc2cc(C(=O)NCc3n[nH]c4nccn34)[nH]c2cc1F
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Fc1cnc2nc(Nc3ccc4cc5c(cc4n3)NNO5)[nH]c2c1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Nc1n[nH]c2c(=O)[nH]c(Nc3cnc4ccc(F)cc4c3)nc12
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N COCc1n[nH]c(Nc2nc(F)c3c(n2)[nH]c2ccc(C)cc23)n1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N O=C(NNc1nc2[nH]c3ccccc3n2n1)Nc1ccc(F)cc1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Cc1cc(F)cc(-c2n[nH]cc2NC(=O)c2nnc3[nH]ccn23)c1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Fc1cc(Nc2nc3ncccc3[nH]2)cc(OCc2cn[nH]n2)c1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Nc1nc(F)c2nc(-c3ccnc(NCc4ccco4)c3)[nH]c2n1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Nc1nn(-c2cc(O)cc(F)c2)c2cccc(-n3ncnc3N)c12
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N CC(=O)c1c[nH]c(-n2cc(-c3ncc[nH]3)c(-c3cn[nH]c3)n2)c1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N CNc1nccc2c1[nH]c1ccc(OC(F)c3nc(N)n[nH]3)cc12
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Cc1cc(F)c(-c2nc3ccc(Nc4cnnc(N)n4)cc3[nH]2)o1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Fc1cc2c(NCc3cn[nH]c3)ccnc2n1Cc1ccn[nH]1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Nc1cc2nc3[nH]c(=NCO)cc(-c4ccncc4F)n3c2cn1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Fc1ccc2[nH]nc(NCc3noc(Nc4ccccc4)n3)c2n1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N O=C(NCc1cc[nH]c1)Nc1nc2cc3ccc(F)cc3nn2n1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Nc1ncnc2nc3cc(F)nc4c3c(c12)n1n4C(CO)CC1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Cc1[nH]nc2[nH]cc(C=NNC(=O)c3c[nH]c(C=CCCF)n3)c12
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N CCc1nnc(N(C)C(N)=NC(=O)c2cc3ccc(F)cc3[nH]2)[nH]1
n1(nnc2c1nc(nc2c1occc1)N)Cc1ccc(c(c1)F)N Cc1cc2nn3c(N)cnc3c(=O)n2c(Nc2ccc(F)cc2)n1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N C=C(C)c1cc(C(=O)Nc2ccc3nc(Br)ccc3c2)[nH]c1C
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N C=Cc1c(C)cc(CC(=O)Nc2cc(Br)n[nH]2)c2ccccc12
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N O=C(CCCc1c[nH]c2ccc(Br)cc12)N1CCc2c[nH]cc21
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CCN=c1cc(C(=O)Nc2cccc(Br)c2)[nH]c2ccccc12
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N Cc1cc(C)cc(-c2cc(C(=O)Nc3ccc(Br)cc3)[nH]n2)c1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N Cc1ccc(C)c(NC(=O)c2cc(-c3ccc(Br)cc3)[nH]n2)c1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CC1(C)Cc2[nH]c3cc(Br)cc(CNc4cccnc4)c3c2O1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CC(=NNC(=O)c1cccc(Br)c1)c1cc2ccc(C)cc2[nH]1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N Cc1cc(Nc2ccc(Br)cc2)cc2c(CO)nn(C3CC3)c12
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CNC(C)=Nc1c[nH]c2c(C=CCO)c(Br)c3ccccc3c12
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CC(Cc1nc2ccc(Br)cc2[nH]1)Nc1ccc2c(c1)CCO2
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CC=Cc1[nH]cc(C)c1NC(=O)Cc1c[nH]c2ccc(Br)cc12
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N Cc1ccc(NC(=O)c2[nH]nc(C)c2-c2ccc(Br)cc2)cc1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CC(c1cccc(Br)c1)N(C)C(=O)Nc1ccc2[nH]ccc2c1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CCc1cc(NC(=O)N(C)c2ccc(Br)cc2)c2c[nH]cc2c1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CC(Cc1[nH]c2cccc3c2c1C(=O)N3)c1cc(Br)n(C)c1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N Cc1ccc(NCCBr)c(C(=O)Nc2ccc3[nH]ccc3c2)c1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N O=C(Nc1ccc2cc(Br)cc(C3CCC3)c2c1)c1cc[nH]n1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N Cc1cc(C(=O)Nc2ccc(Br)cc2-c2ccc(C)[nH]2)ccn1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CNCc1[nH]c(=Nc2ccc(Br)c3ccccc23)oc1C(C)C
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CCc1ccc(C)c(C)c1NC(=O)c1nc2[nH]ccc2cc1Br
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N Cc1cc(=O)[nH]nc1Cc1ccccc1Nc1cccc(Br)c1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N Cc1cc2c(C(=O)Nc3cccc(Br)c3)cc(C3CC3)nc2[nH]1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CCc1cc2cc(NNC(=O)c3ccncc3)ccc2cc1Br
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N O=C(CBr)Nc1cccc(-c2ccc3[nH]c(C4CC4)nc3c2)c1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N Cc1n[nH]c(-c2ccc3cc(Br)ccc3c2)c1C(=O)NC1CC1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CC(=N)C(=O)Nc1ccc(Cc2ccc3[nH]c(Br)cc3c2)cc1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N O=C(NNc1cccc2ccccc12)Nc1cccc(CBr)c1
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CCNc1cccc2[nH]c(CO)cc(=Nc3cccc(Br)c3)c12
n1c(nc(c2c1c1c(C2)ccc(c1)C(C)C)c1ccc(o1)Br)N CCc1cc(Br)c(NC(=O)Nc2cccc3[nH]ccc23)cc1C
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 C=CC(=C)c1cc(-c2ccc3oc(=O)[nH]c3c2)[nH]n1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=c1[nH]c2ccc(C=NNc3ccccc3)cc2o1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 Oc1ccccc1Oc1cccc(-c2nnc[nH]2)c1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 Oc1ncncc1C=COc1c[nH]c2ccccc12
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 CC(=O)Nc1ccc2oc(-c3ccc[nH]3)nc2c1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 Oc1[nH]ccc1-c1ccc(Oc2cnccn2)cc1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 C=CC(=O)Nc1[nH]ncc1-c1cccc2ccoc12
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 Cc1oc2cc(NC(=O)c3cn[nH]c3)ccc2c1C
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=C(NN=Cc1ccoc1)c1cc2ccccc2[nH]1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=COc1ccc(N=c2[nH]c3ccccc3[nH]2)cc1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 CNC(=O)Nc1ccc2nc3occc3cc2c1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=C(O)Nc1cccc2c1ccn2Cc1cc[nH]c1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=c1c2ccccc2[nH]c(=Nc2ccccc2)n1O
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=c1[nH]c2ccccc2cc1Nc1ccnc(O)c1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 COCC(=O)Nc1cnc2[nH]c3ccccc3c2c1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 OC(c1cc(-c2nc3cnccc3o2)c[nH]1)C1CC1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=c1[nH]ncn1-c1ccc(Oc2ccccc2)cc1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=c1[nH]cccc1-c1nccn1-c1ccc(O)cc1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 Cc1cc(NC(=O)c2ccc3oc(C)cc3c2)[nH]n1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 CCCc1c[nH]c(-c2nc3cc(C)[nH]c(=O)c3o2)c1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=C(Nc1ccccc1)Nc1noc2ccccc12
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 NC(c1ccc2onnc2c1)c1cc2c(o1)CCC2
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 Oc1ccc(-c2cnc(-c3ccncc3)[nH]2)cc1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=C(Nc1ccccc1O)c1cnc2ccccn12
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 c1cc2c(cc1Oc1cnc3[nH]ncc3c1)COC2
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=C(Nc1ccccc1O)c1ccc2cn[nH]c2c1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 Cn1c(=O)[nH]c2cc(Oc3ccc(N)cc3)ccc21
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 Cc1ccc(CNC(=O)c2nc3ccccc3[nH]2)o1
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 O=C(NCc1cc[nH]c1)Nc1coc2ccccc12
c1c(nc(c(c1c1occc1)C#N)N)c1ccco1 Cc1nc(-c2cc(O)cc3cc(O)c(C)cc23)n[nH]1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1cc(-n2ccc3c(C(=O)Nc4ccc(CN)nc4)n[nH]c32)no1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Nc1nc2ccc(Cc3ccnc(Oc4cnnc(O)c4)c3)nc2[nH]1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O CNCC(=O)Nc1nc2cc(-c3c[nH]cc3-c3nc[nH]n3)ccc2o1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1cc(-c2cc(C(=O)Nc3ccc4[nH]ncc4c3)[nH]n2)nc(O)n1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1cc(Cc2c[nH]nc2NC(=O)c2ccc(-c3cc[nH]n3)[nH]2)no1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1cc(-n2[nH]c3nc(Nc4cc[nH]c4)[nH]c3c2=O)ccc1NC=O
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Nc1cnc(C=Cc2nc3cc(O)ccc3o2)nc1Nc1ncc[nH]1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1cnc2nc(Nc3cc(-c4ccc(O)c(O)c4)n[nH]3)nn2c1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1ncc(-c2nc3c(cc(C)n3-c3nc[nH]n3)c(=O)[nH]2)cc1CO
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1c(C=Cc2nnc(N)o2)oc2cc(Nc3nc[nH]n3)ccc12
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O O=C(Nc1ccc(CCNc2ncnc3[nH]cnc23)cc1)c1c[nH]o1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Nc1cc(-c2cc(-n3cc(-c4ccc(O)c(N)c4)cn3)ncn2)on1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O COc1ccc(Oc2nnc(-c3cnc(-c4cc(C)n[nH]4)[nH]3)[nH]2)cc1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O O=C(Nc1ccc2cc[nH]c2c1)C(=O)Nc1cnn(-c2cc[nH]n2)c1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O O=C(Nc1nccc(CO)n1)Nc1ncnc2[nH]c3ccccc3c12
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cn1c2ccccc2c2c(C(=O)NNc3ccn[nH]3)n[nH]c(=O)c21
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O CCc1cc(-n2nnn3c4nc(N)ccc4c(=O)nc23)cc(C)c1O
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1nc2c(N)nc(-c3ccc(Cn4nccc4CCO)o3)nc2[nH]1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O CNOc1ccnc(-c2nc3ccc(=O)[nH]c3n2-c2c[nH]nc2C)c1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O O=C(Nc1cnc(Nc2cn[nH]c2)nc1O)c1ccc2cc[nH]c2c1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O O=C(Nc1ccc(O)cc1)Nc1ccnn1-c1ccc2nc[nH]c2n1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1cccc(NC(=O)c2c(CO)cc3nnc4nc(N)[nH]c2n34)c1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Nc1cc(-c2nc(-c3cccc(CO)c3)no2)cc(-c2nnc[nH]2)n1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O CCc1cc(-c2nc(N)nc(-n3c(=O)oc4ccc(C)cc43)n2)[nH]n1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1cc(C)cc(NC(=O)c2coc(-c3n[nH]c4nc(N)nn34)c2)c1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O NNc1nc(COc2cccc3ccoc23)ccc1-c1ncn[nH]1
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O CN=CC(=O)c1c(-c2ccc3oncc3c2)nn(-c2ncc[nH]2)c1N
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O COc1ccc2c(c1)[nH]c1cc(C(N)=Nc3ncncn3)ncc12
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O C=NNC(=O)c1cc2cc(NC(=O)NCc3cc[nH]n3)ccc2n1C
c1c(ccc(c1)CCNc1nc(n2c(nc(n2)c2ccco2)n1)N)O Cc1ccc2nc(NNC(=O)c3n[nH]c4cocc34)n(C3CC3)c2n1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C C=C(C)SCc1nnc2sc3ccccc3n12
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CCSc1nnc(-n2ccc3ccccc32)s1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CN(c1ccsc1)c1ccnn1-c1ccsc1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C C=CCSc1nnc2sc3ccc(C)cc3n12
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CCCCSc1nnc2sc3ccccc3n12
n1c(nc(c2c1ccs2)c1nccs1)C(C)C C=C(CS)Cc1nnc2sc3ccccc3n12
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CCCSCc1nnc2sc3ccccc3n12
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CSc1ccn(-c2ncnc3sc(C)cc23)c1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1cnc(Sc2nc3ccccc3s2)n1C
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1ccc2c(c1)sc1nnc(SC(C)C)n12
n1c(nc(c2c1ccs2)c1nccs1)C(C)C c1ccc(Sc2nnc(-n3cccc3)s2)cc1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1ncsc1CSc1ccn2ccnc2c1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1csc2nnc(CSc3ccccc3)n12
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CCc1csc(-n2c(S)nc3ccccc32)n1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1nc(Sc2nccs2)n2cccc2c1C
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1nn(C)c2nc(C=Cc3ccsc3)sc12
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1cnc(Cc2csc(-n3cccc3)n2)s1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C SCCc1cnn(-c2nccc3cscc23)c1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CN(C)c1nsc2nccc(-c3ccsc3)c12
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CCSc1nc2c(cnn2-c2ccccc2)s1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CCCc1ccc(-n2nc(C)c3scnc32)s1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C c1ccc2nc(CSc3nncs3)ccc2c1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1ccn2nc(SCc3ccsc3)nc2c1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1ccc(CSc2nnc3ccccn23)s1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CCC(C)c1cc(-c2nnc3sccn23)cs1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CSc1ccc(Cn2cnc3cnccc32)s1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CCN(C)Sc1ccc2nc3sccn3c2c1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C C=CC(=C)c1ccc(-c2cn3cnnc3s2)s1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C CNCc1cc2c3ccccc3sc(=S)n2n1
n1c(nc(c2c1ccs2)c1nccs1)C(C)C Cc1ncc(-c2ncncc2-c2ccsc2)s1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCn1[nH]c(=Nc2ccc(OC)cc2OCCc2cc[nH]c2)[nH]c1=O
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC COCCN(CC(C)NC(N)=O)c1cc2c(nn1)oc1ccccc12
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC Cc1ccc(O)c(OCCNC(=O)c2ccc(-c3nnn[nH]3)cc2)c1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CC=Cc1cnc(C(C)C)c2c(O)nc3ncc(C(N)=O)c(=O)n3c12
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCC(CC)Oc1cc(C(=O)N=c2[nH]c(=O)c3cc[nH]c3[nH]2)ccn1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCN(C)c1n[nH]c2[nH]c(=O)c(NC(=O)c3ccc(OC)cc3)cc12
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCOc1ccc(-n2nc(-c3cc(NC=O)[nH]n3)cc2C(C)O)cc1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC Cc1cc(-c2cc(C(=O)Nc3nn(C)c(=O)cc3C)[nH]n2)ccc1O
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CC(C)(C)c1noc(CNC(=O)c2cc3cnc(CCO)cc3[nH]2)n1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CNNC(=O)COc1ccccc1-c1noc(C=Cc2cc[nH]c2)n1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCc1ccc(-c2nnc(C(=O)NN=Cc3cccc(C)c3O)o2)[nH]1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC C=Nc1nccn1CC(=O)Nc1c[nH]c(C(=O)c2ccc(O)cc2)c1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCNC(=O)CNC(=O)CCc1ccc2oc(-c3ccn[nH]3)cc2n1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC O=C(CO)NCCOc1cc(Nc2ncc3ccccc3n2)ccn1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC NC=Cc1ccnn1C(=O)C(=Cc1cn[nH]c1)Oc1ccc(O)cc1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCc1ncnc(NC(=O)Nc2ccc3cc(O)c(OC)cc3c2)n1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CC(COc1ccccn1)NC(=O)Nc1ccc2c(c1)c(O)nn2C
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC O=C(C=Cc1ccc(O)cn1)Nc1cc(C=CCc2ncc[nH]2)on1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCOCCOc1ncnc(-n2ccc3[nH]c(=O)c(CC)cc32)c1N
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC COc1ccc(NC(=O)CCc2ccc3[nH]c(NC=O)nc3c2)cn1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC O=C(Cn1ncc(C(=O)Nc2cccc3ccccc23)n1)NCCO
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC COc1cc(C(=Nc2cn[nH]c2)NCc2nc(C)c(C)o2)ccc1O
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC Cc1cc(NC2CC2)nc2nc(-c3ccc(O)c(OCCO)c3)nn12
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC COc1cccc(-n2c(C)n[nH]c2=NC(=O)Nc2ccc(O)cc2)c1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCOc1ccc(NC(=O)Nc2cc3cnn(CC)c3[nH]c2=O)cc1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCc1cc(CNC(=O)c2ccc(NC(=O)c3ccoc3)cn2)[nH]n1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC CCOC(=O)c1cc(CC(=O)Nc2cccc(-n3ccnc3)c2)[nH]n1
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC C=C(OC)c1cc(NC(=O)Cn2ncncc2=O)cc2cc(C)[nH]c12
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC O=C(NCCCc1ccc(-n2ccnn2)cc1)c1c(O)ccnc1O
c1c(nc(nc1c1occc1)N)C(=O)NCc1cccc(n1)COC Cn1ncnc1Nc1ccc(OCc2ccc(NC=O)cc2O)cc1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N O=C(Oc1cccc(-n2cccn2)c1)C(CBr)=NNc1ccc[nH]c1=O
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N C=C(O)C(=CC)n1nnc2cc(Br)c(Cn3c(C)cc(=O)[nH]c3=O)cc21
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N Oc1nc2c(Br)cnn2c2ncnc(CCCOC3CCC(O)CC3)c12
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CCc1cc(NC(=O)COC(=O)c2[nH]cc(C#N)c2Br)n2nccc2c1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N COC(=O)c1[nH]ncc1N(C)C(=O)c1[nH]ncc1-c1ccc(Br)cc1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N COC(=O)c1c[nH]c(C=C(Br)CC(=O)Nc2nncc3ccccc23)n1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CCOc1ccc2[nH]c(=NC(=O)C=Cc3cc(=O)[nH]c(Br)n3)n(C)c2c1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CN(CNC(=O)c1ccnc2oc(C3CC3)nc12)C(=O)c1cc(Br)c[nH]1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N Cc1cc(C(=O)O)n(-c2ncc(C(=O)Nc3ccc(Br)nc3)cc2C)n1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N COc1ccc(NC(=O)Nc2ccccc2-n2ncn(C)c2=O)c(Br)c1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N C=CCNC(=O)c1noc(-c2cccc(Br)c2)c1C(=O)Nn1ccnc1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CCNC(=O)COc1ccc(Br)c(N=Cn2ncc3ccc(O)nc32)c1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N O=C(Nc1ccc(-n2cncn2)cc1)C(=O)Nc1ccccc1OCBr
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N Cc1n[nH]c(C)c1Oc1cc(NC(=O)Cn2cccc(Br)c2=O)ccn1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N COc1ccc(NNC(=O)COc2ncc(Br)n3cc(C#N)cc23)cc1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N Cc1cc(C(=O)N(C)CC(=O)N=c2[nH]c3cc(C)c(Br)cc3[nH]2)on1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CCOc1cc(NC=NC(=O)c2nc(Br)cc3nc[nH]c23)ccc1OC
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N O=C(NN=Cc1c2n(c3ccoc13)CCN2CCO)c1cncc(Br)c1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CNC(=O)Oc1ccc(-n2nncc2C(=O)Nc2cccc(Br)c2)cc1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CN(C)C(=O)c1nn(-c2ccc(Br)cc2)c2cc(NNC(=O)O)ccc12
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N COc1cc(Br)cnc1N(C)Cc1ccc2[nH]c(C3COCO3)nc2n1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N Cc1c(Br)c(=O)n(N=Cc2cc(O)ccc2O)c2nc(N(C)C)ncc12
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CCCCOC(=NC(=O)c1cc2nnc(Br)cc2o1)NCc1cc[nH]c1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CC(=CC(=O)NCc1ccnc(NC(=O)Br)n1)c1nc2ccccc2o1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N O=C(CCc1cnn(Cc2ccco2)c1)Nc1cnc(C=CBr)[nH]c1=O
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CN(Cc1ccn[nH]1)C(=O)Nc1cccc(Br)c1Oc1ccc[nH]c1=O
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N O=C(CNC(=Nc1ccccc1)n1nc[nH]c1=O)Oc1cccc(Br)c1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N Cn1cc2nc1C(OCNC(=O)Cc1nc(=O)c3cccc(Br)c3[nH]1)=C2
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N O=C(CCOc1ccccc1Br)N=c1[nH]nnn1-c1cccc(CO)c1
n12c(nc(n1)c1oc(cc1)Br)cc(C(=O)N1[C@@H](COC)CCC1)cc2N CC1(C(=O)NCc2nc(-c3ccn[nH]3)no2)OCCc2cccc(Br)c21
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=c1[nH]c(-c2ccc(Cl)cc2)cc2nn(Cc3cc[nH]n3)cc12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=c1nc2[nH]c(CNc3ccccc3Cl)nn2c2ccccc12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=C(NCc1cnc2c(Cl)cccn12)c1cc2cnccc2[nH]1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=c1nc2nc(Nc3ccc(Cl)cc3)[nH]n2c2ccccc12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Cn1cc(N=c2[nH]c(=O)c3ccccc3[nH]2)c2c(Cl)ccnc21
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=C(N=c1ccc2ccc(Cl)cc2[nH]1)c1cnn2cc[nH]c12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Cc1nccn1C(C)c1nc2c(=O)[nH]c3cc(Cl)ccc3c2[nH]1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl OCc1ccc(-c2nnc3cc(Cl)c(-c4ccncc4)cn23)[nH]1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Oc1cccc2c(-c3ncc(-c4ccnc(Cl)c4)[nH]3)cnnc12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Cc1cc2oc(N=C(N)c3cccc(Cl)n3)cc2c2nccn12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl OCc1ccnc(N=c2[nH]nc3c(=CCl)c4ccccc4n23)c1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Oc1ccc(-n2cnc(Nc3cc4[nH]ccc4cc3Cl)n2)cc1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=C(C=Cc1c[nH]c(-c2n[nH]c3c[nH]n23)c1)c1ccc(Cl)cc1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl NCc1ccc2c(=O)nc(-n3ncc4cc(Cl)ccc43)[nH]c2c1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Oc1ccc(Cl)cc1CNc1ncnc2c1nc1ccccn12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=C(Cn1cccc1Cl)Nc1ccc2nc3ncccn3c2c1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Oc1ccc(-n2ccc(Cn3cnc4ccc(Cl)nc43)c2)nc1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl CC(=O)Nc1nn(-c2nc3ccccc3[nH]2)c2ccc(Cl)cc12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl C=NC(=CC)N=c1[nH]c(=O)[nH]n1-c1cccc2c(Cl)cccc12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=C(Nc1cnc(Cl)c2ccccc12)c1ccn2cnnc2c1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl CC(C=Cc1cccc2n[nH]c(=NC(=O)c3ccc[nH]3)n12)=CCl
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl ON=C(c1ccc(Cl)cc1)c1n[nH]c2nc3ccccc3nc12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Cn1nc(CO)cc1Cn1cnc2c3ccc(CCl)cc3[nH]c21
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Cc1cc(Cl)ccc1-c1ncnc2c1c(=O)[nH]c1nccn12
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Clc1ccc2nc(-c3noc(CNc4ccccc4)n3)[nH]c2c1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=Cc1ccc(NC(Cl)=Nc2nc3cccc4ncn2c43)cc1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=C(N=c1[nH]cc(Cl)n1-c1ccccc1)c1cc(C2CC2)[nH]n1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl CCn1c(-c2cc3ncccc3c(=O)[nH]2)nc2nc(Cl)ccc21
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl Cc1cc2ccc(Cl)cc2n1-c1cc(NCC2CN=CO2)[nH]n1
c1(ccc2c(c1)n1n(c(n2)N)nc(c1=O)c1ccc(cc1)C)Cl O=C(Nc1ccnc2ccc(Cl)cc12)c1ccnc2ccnn12
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC C=C1OC=CC=C1Cc1onc2nc(N(CC)C(C)C)[nH]c(=O)c12
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CCN(CC)c1nc2c(C=CC3=CCOCC3C)noc2c(=O)[nH]1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CCOC(=CC(=O)OC)c1nc(N2CCC(C)C2)c2cc[nH]c2n1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC Cc1nnc(CCC(=O)Nc2ccc(OC3C=CCC3)nc2C)o1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CCC(Oc1ccc2cnn(CC)c2c1)C(=O)NC1=NOC(C)C1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CN=Nc1[nH]c2cc(O)ccc2c1CCCC(=O)N1CCOCC1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC COc1ccc(OCc2nnc(C3NC4CCCN3C4C)o2)cc1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC COc1ccc(C=NNC(C)c2nc(C3=CCOC=C3)no2)cc1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CCOc1ccc(C=CC(=O)N=CNc2ccc(C=O)nc2)nc1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC C=C(C=O)C(=CC)OC(=O)NCc1cn(-c2ccncc2)nc1C
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CN=CN=C(Nc1cc(OC)ccc1OC)c1ccc(OC)cn1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC Cc1nc(C)c(CNCc2nc(C=O)c(N3CCCC(C)C3)o2)o1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CCc1nccn1-c1ccc(NC(=O)N(C)C(C)C(=O)OC)cc1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC COc1ccc(Nc2nnc(C)nc2OCCC2CCCO2)cc1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CCOC(=O)C=NNCc1ccc2oc(N3CCCCC3)nc2c1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CCN(CC)C(=O)Nc1ccccc1OC(=O)c1ccc(C)nn1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CC(=NOCC(=O)C#N)c1cccc(NC(=O)c2ccn(C)c2)c1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CC(=CC=O)C(=O)Nc1ccc(N=Cc2ccnn2C)c(C)c1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC Cc1n[nH]c(C)c1CC(=O)N=c1cc(O)cc(C)n1C1=COCC1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CN(C(=O)c1ccc(O)cn1)c1ccc(C=NOCCC#N)cc1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CC(=NN(C=O)c1ccc(NC(=O)c2ccoc2C)cc1)N(C)C
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CN(CCc1nc2ccccc2[nH]1)C(=O)CCC(=O)OCCC#N
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC COCc1nc2cc(C(=O)N(C)CC3=CCNN=C3C)ccc2o1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC COc1ccc(C)c(NC(=O)c2nc(C)n(C3=CCOC=C3)n2)c1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC Cc1ccc(C#N)cc1NC(=O)COc1ccc(C=CC=O)nn1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC C=NN(C)c1cc(=O)occ1C(=O)NN=CCc1ccc(C)cc1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC COc1cc(C#N)ccc1N(C)C(=O)Cc1coc(NC2CC2)n1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC CC(=O)Nc1ccc(-c2nnc(CC(C)=CC(=O)N(C)C)o2)cc1
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC Cc1c(C(=O)NN=C(C=CC2=CCOC2)c2ccoc2)cnn1C
c1(nc(nc(c1)NC(=O)C)c1ccc(o1)C)N1[C@H](CCC1)COC COC(C)CN(Cc1ccoc1)C1CCC(n2nc[nH]c2=O)C1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 Cc1nn2c(C=CC=Cc3cnc(N(C)C)[nH]3)nnc2[nH]1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCCc1c(-n2ccc(NCc3ncc[nH]3)n2)nnn1C
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCC(CC)n1cc(NCCc2nnc3[nH]cnn23)cn1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 C=CCc1cnn(-c2nnc(Cc3nc(C)n[nH]3)[nH]2)c1C
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 Cc1n[nH]c2c1c(NCCCn1ccnn1)nn2C(C)C
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCCCNCc1ncnc2cnn(Cc3nc[nH]n3)c12
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 Cc1n[nH]c(NCc2nccn2CCc2cnn(C)c2)n1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CN(C)c1ccc(-n2cnnc2CNc2c[nH]nn2)cc1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCc1cc(CNc2cc(-n3ncnc3C)ncn2)n[nH]1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CC=C(C)C=Cn1nc(NCc2cnc[nH]2)n2ncnc12
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 Cc1cc(NC(C)c2nnnn2-c2ncc[nH]2)c(C)n1C
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCc1n[nH]c(NCCCc2cc(C)cc3nnnn23)n1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCC(C)CNc1nncnc1-n1nc(C)c2[nH]ncc21
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCC(C)c1[nH]nnc1C(C)Nc1cnn2ccnc2n1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CNC(C)c1cc(CNc2cccc3nnnn23)nn1C
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCCCCCc1nc(-c2nnc3[nH]nnn23)[nH]c1CC
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 Cc1n[nH]c(C)c1-c1n[nH]c(-c2cncc(N(C)C)n2)n1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCN(C)c1nc(CNc2ccn[nH]2)c2c(ncn2C)n1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCn1ncc(CCNCc2nn3c(C)nnc3[nH]2)c1C
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 Cc1cc(CN(Cc2n[nH]c(C)n2)Cc2cnc[nH]2)n[nH]1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 C=C(C)C=Cc1n[nH]c(-c2n[nH]c(-c3nccn3C)n2)n1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CC(CCNc1nnc2cn[nH]c2n1)Cc1cnccn1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 Cc1ccc(NC(C)c2nnnn2-c2c[nH]nn2)cc1C
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CN(C)C=Cn1c(N)cn2c(C=Cc3ccn[nH]3)nnc12
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCNc1cn(C(C)C)c2nc(Cn3nnnc3C)[nH]c12
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CC(=Cc1cnn(C)c1)Cn1cnnc1Nc1ccn[nH]1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 Cc1n[nH]c(NC(CCn2cccn2)c2cnccn2)n1
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCc1nnc(CNc2ncc3[nH]c(C)nc3n2)n1CC
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCNc1nc(NCc2ccnn2C)cc2nnc(C)n12
c1(n(c2c(n1)c(nc(n2)CCCCC)N)C)n1nccn1 CCc1ncc(CNc2ncc3nccn3n2)nc1NC
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Nc1cc(C=O)c2n[nH]c(=Nc3ccc4[nH]ccc4c3)n2c1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Nc1ccc2cc3c(=O)[nH]c(=Nn4cccc4)[nH]c3nc2c1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N NCCNc1ncnc2[nH]c(=O)c3c4ccccc4[nH]c3c12
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Cn1cc(-c2cc3ccccc3c(=O)[nH]2)c2c(NN)n[nH]c21
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Cn1cc(NCc2n[nH]c3c(=O)[nH]c4ccccc4c23)cn1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N O=c1[nH]c2ccccc2c(Nc2cn[nH]c2)c1-c1cc[nH]n1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Nc1ncnn1-c1ccc2cc3c(CCO)c[nH]c3nc2c1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Cc1cc2nc3nc4nc(N)[nH]c4cc3nc2cc1CCO
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N NC(=O)Nc1nc2ccc3cc(-n4ccnc4)ccc3c2[nH]1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Nc1cnc2[nH]c3cc(Nc4ccccn4)ccc3n2c1=O
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N CCN1COc2cc3[nH]c4[nH]ccc4c(=NN=CN)c3cc21
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Cc1c[nH]c(=O)c2cc(Nc3nc4ncncc4[nH]3)ccc12
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Nc1nccnc1-n1c(N)nc2c3cc(O)ccc3ccc21
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N O=c1[nH]c2ccc(Nc3cc(-c4cc[nH]n4)ccn3)cc2[nH]1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N NN=C1N=C(Nc2cccc3ccccc23)n2[nH]c(=O)cc21
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Nc1cccc2nc(C(=O)Nc3ccc4n[nH]cc4c3)[nH]c12
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Oc1nncc2ccc(NCc3nc4ccccc4[nH]3)nc12
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N O=CCc1cc(-c2nc3ccc(-c4ccn[nH]4)cc3[nH]2)[nH]n1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Nc1nn2cc[nH]c2c1C(=O)Nc1cnc2ccccc2c1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Cc1nc[nH]c1C(=O)Nc1cccc2cc3cn[nH]c3nc12
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Cc1cc(-n2c(-c3cc[nH]c3)nc3ncc(N)n32)ccc1O
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Nc1ccc(Oc2ccc3c(n2)[nH]c2ccc(N)nc23)cn1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Nc1cccc(-c2[nH]nc3c2cnn3-c2cc(O)ccn2)c1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Cc1nn2c3ccc(NCCN)nc3nc3ccc(=O)c1c32
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Oc1cc(Nc2[nH]ncc2-c2nc3ccccc3[nH]2)ccn1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Cc1nc(O)cc(-c2nc(N)c3[nH]c4ccccc4c3n2)n1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N NC(=O)c1c(-c2ccc3[nH]cnc3c2)cc2nccn2c1N
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N Cc1nnc(-c2cc3cc(-c4cccnc4)[nH]c(=O)c3[nH]2)[nH]1
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N O=C(Nc1ccc2[nH]ccc2c1)Nc1n[nH]c2ncccc12
n12c(nn(c1=O)c1ccc(N)cc1)c(nc1c2cccc1)N COc1cc(Nc2cc(N)c3[nH]ccc3c2)nc2n[nH]cc12
c1cccc(c1)c1nc(nc(n1)N)SCC CCc1csc(=Nc2ccc(NC)nc2)[nH]1
c1cccc(c1)c1nc(nc(n1)N)SCC Cc1csc(CNc2cc(C3CC3)n[nH]2)n1
c1cccc(c1)c1nc(nc(n1)N)SCC CCNCc1cc(N=Cc2cn[nH]c2)cs1
c1cccc(c1)c1nc(nc(n1)N)SCC C#Cc1cnc(Nc2nc(CC)c(C)[nH]2)s1
c1cccc(c1)c1nc(nc(n1)N)SCC C=CCNc1ccc(-c2cc(S)[nH]n2)cn1
c1cccc(c1)c1nc(nc(n1)N)SCC CC=CSc1ncc(N)c(-n2cccc2)n1
c1cccc(c1)c1nc(nc(n1)N)SCC C=Nc1cc(Sc2nccn2C)ccc1N
c1cccc(c1)c1nc(nc(n1)N)SCC Cc1sccc1NCc1nc(C2CC2)n[nH]1
c1cccc(c1)c1nc(nc(n1)N)SCC CNCc1csc(Nc2cncc(C)c2)n1
c1cccc(c1)c1nc(nc(n1)N)SCC Cc1cc2sc(C=NN(C)C)cc2c(N)n1
c1cccc(c1)c1nc(nc(n1)N)SCC CNC(C#N)CNc1nc2ccccc2s1
c1cccc(c1)c1nc(nc(n1)N)SCC Cc1nc(C=Cc2cnc(N)c(C)n2)cs1
c1cccc(c1)c1nc(nc(n1)N)SCC CN=CN(C)Cc1cc2ccnc(N)c2s1
c1cccc(c1)c1nc(nc(n1)N)SCC Cc1[nH]nc2nc(NC3CCSC3)ccc12
c1cccc(c1)c1nc(nc(n1)N)SCC Cc1cc(N=C(N)c2cnccn2)sc1C
c1cccc(c1)c1nc(nc(n1)N)SCC CCSc1ccccc1NCc1nc[nH]n1
c1cccc(c1)c1nc(nc(n1)N)SCC CSC(N)=NN=Cc1ccc2cc[nH]c2c1
c1cccc(c1)c1nc(nc(n1)N)SCC CSc1cc(C)cnc1NCc1ccn[nH]1
c1cccc(c1)c1nc(nc(n1)N)SCC CCCc1c(C)n[nH]c1SCc1ncc[nH]1
c1cccc(c1)c1nc(nc(n1)N)SCC N#CCSc1ccc(Nc2ncc[nH]2)cc1
c1cccc(c1)c1nc(nc(n1)N)SCC CCNc1ccccc1Sc1nc(C)n[nH]1
c1cccc(c1)c1nc(nc(n1)N)SCC Cc1cc(CCc2c(C)ncnc2S)n[nH]1
c1cccc(c1)c1nc(nc(n1)N)SCC Cc1cc(CNC(=N)c2cn[nH]c2)c(C)s1
c1cccc(c1)c1nc(nc(n1)N)SCC CCSc1nnc(-c2ccc[nH]2)n1C1CC1
c1cccc(c1)c1nc(nc(n1)N)SCC Cc1n[nH]cc1-c1nsc(CCC2CC2)n1
c1cccc(c1)c1nc(nc(n1)N)SCC CCc1cc(Nc2nccc(C)c2S)n[nH]1
c1cccc(c1)c1nc(nc(n1)N)SCC CC=C(C)C=Cc1nn(C)c2nc(N)sc12
c1cccc(c1)c1nc(nc(n1)N)SCC CC(=N)NCCSc1nc2ccccc2[nH]1
c1cccc(c1)c1nc(nc(n1)N)SCC CNc1cc2c(cc1C)c(NC)nn2C
c1cccc(c1)c1nc(nc(n1)N)SCC CNc1cc(NCc2ccc(S)cc2)[nH]n1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 CC=C(F)c1cc(O)ccc1NC(=O)c1nn2c(c1F)CSCC2
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 Cc1ccc(NC2=NC(=O)C(=Cc3cc(F)cnc3F)S2)c(O)c1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 COC(=O)c1ccc(NC(=S)Nc2cc(F)cc(F)c2C#N)cc1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 C=CCNC(=NS(=O)(=O)CC(F)F)Nc1cccc2ccccc12
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 CCC1CNc2c(sc(=Nc3ccc(OC(F)F)cc3)[nH]c2=O)C1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 O=C(c1cc(F)cc(F)c1CO)N(C1=CCSC=C1)c1ccn[nH]1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 O=C1N=C(Nc2cccc(-c3cccc(O)n3)c2)SC1=CC(F)F
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 CC(C)(C)Cc1ncc(C(=O)Nc2c(F)ccc(NC=O)c2F)s1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 O=C(NN=C1NCCS1)c1cc(F)cc(Oc2ccccc2F)c1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 N=C1CSC(=NC(=O)c2ccc(F)cc2Oc2cccc(F)c2)N1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 N=C(S)C(=NCF)C(=O)Nc1cc(F)ccc1Oc1ccccc1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 Cc1c(F)cc(NC(=S)ON=C2C(=O)Nc3ccccc32)cc1F
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 N=C1C=c2cc(N=CSc3ccc(OC(F)F)cc3)c(=O)[nH]c2=C1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 CNC(=O)Sc1ccc(F)cc1NC(=O)Nc1ccc(F)cc1C
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 O=C(N=C1NNCCS1)c1cc(F)cc(F)c1Oc1ccccc1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 Cc1ccc2c(c1)N=C(NS(=O)(=O)c1ccccc1C(F)F)NC2
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 C=C1N=C(SCc2cc3cc(F)cc(F)c3[nH]c2=O)N(CC)C1=O
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 O=[SH]C1(F)CCCC(NC(=O)Nc2cnc3ccc(F)cc3c2)C1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 C=CC=CCOc1cc(N=c2[nH]c(=O)c(C#N)c(F)s2)ccc1F
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 Cc1ccc(S(=O)(=O)NN=CC(F)=CC=Cc2cc[nH]c2)c(F)c1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 CCN1CCc2nc(COC(=O)Nc3cc(F)ccc3F)sc2C1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 Cc1c[nH]c(CN2CCc3cc(NS(C)(=O)=O)cc(C(F)F)c32)c1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 C=Nc1snc(C2CC2)c1C(=O)Nc1ccc2c(c1)CC(F)(F)O2
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 Cc1ccc(NC(=O)Nc2cc(F)c(F)cc2SCC#N)cc1O
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 O=S(=O)(NCc1cc[nH]c1)c1cc(N2CCCCC2)c(F)cc1F
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 CC1CCSCc2c1nn(C)c2NC(=O)c1cc(F)ccc1O
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 CSC(=NC(=O)Nc1ccc(OCc2ccccc2)cc1F)NF
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 Nc1ccc(F)cc1C(=O)N=c1sccn1CC1=C(F)COC=C1
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 CN1CCCNc2cc(S(=O)(=O)Nc3cc(F)ccc3F)ccc21
c1(cc(c(c(c1)F)NC(=O)CC(C)(C)C)F)C(=O)Nc1sccn1 CC(=NS(=O)(=O)Nc1ccc(C(F)F)cc1)Nc1ccc(C)cc1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CN=c1[nH][nH]c2ncc(C(=O)NCCCc3ccc(F)cc3)cc12
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C N#CCNCc1cnc(C(=O)Nc2cccc3cc(F)ccc23)[nH]1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CC(C)(O)c1nc(N2CC#Cc3c[nH]cc3C2)c2ncc(F)cn12
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Nc1ccn(-c2ccc(F)nc2)c(=Nc2ccc(CO)cn2)c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C O=C(CNc1cccc(-c2ccc(F)cc2)c1)N=c1[nH]cn[nH]1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Cc1c[nH]c2ccc(F)c(CN3CCc4nc(N)[nH]c(=O)c4C3)c12
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CCc1n[nH]c(-c2cc(CNC(=O)c3cc[nH]c3)c(F)cc2C)n1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CCNC(=O)NC(Cc1ncc[nH]1)c1cnc2ccc(F)cc2c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Cc1cc(NC(=O)NCC=Cc2cn3cc[nH]c3n2)ccc1F
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C C=C(C)c1cc(=N)c2c(N)ncnc2n1-c1ccc(OC)c(F)c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CNc1cc(NC(C)=O)cc(N=c2[nH]c3ccccc3cc2F)n1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C NNC(=O)c1cnn(C(Cc2ccc(F)cc2)c2ccncc2)c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Cc1cc(Cc2ccc(F)c(C(=O)Nc3ccc(=N)[nH]c3)c2)[nH]n1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CCc1ccc(CNC(=O)Nc2nc3nc(c[nH]3)c2=C(C)F)cc1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CNc1cc(-n2ncc(C(N)=O)c2Cc2ccc(F)cc2)ccn1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Cn1cc(C(N)C2=CC(O)(F)C=C2)c(-c2nc3ccccc3[nH]2)n1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CCc1ccc(F)c(-c2cc(-n3ncc(CC(N)=O)c3C)[nH]n2)c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Oc1ccccc1C=CCNCc1nc(-c2ccnc(F)c2)n[nH]1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CCNCc1nc(C)cn1CC(=O)Nc1cccc2[nH]cc(F)c12
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Cc1c(N)ncn1CC(=O)Nc1cc(C#N)c2ccc(F)cc2c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C NCc1ccnc(Oc2cc(F)cc(NCc3ncc[nH]3)c2)c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C O=C(Cc1ccn[nH]1)Nc1ccc(CNc2ccncc2)c(F)c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C O=C(Nc1ccn[nH]1)C(=Cc1c#cccc1)Nc1ccc(F)cn1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C CCc1cccc(CNN=c2[nH]nc(-c3ccc(O)c(F)c3)[nH]2)c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Cc1n[nH]c(C(=O)Nc2ccc(-c3ccc(C#N)[nH]3)c(F)c2)c1C
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C C=CCc1ccc(NC(=O)NCc2ncn[nH]2)c2ccccc12
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C O=C(NCc1cccnc1)c1ccc(CNc2cn[nH]c2)c(F)c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Cc1c(C(=O)NCc2ccncc2)nc(N)n1-c1cccc(F)c1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Nc1cn(NC(=O)c2cccc(CCc3ccccc3F)n2)cn1
c12n(c(nc1c(nc(n2)C#CC(O)(C)C)N)c1cc(F)ccc1)C Nc1ccc(C=CCc2nc(Cc3ccc(F)cc3)n[nH]2)cn1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1cc(-c2c(C(N)=O)cc3c(c2O)CN(C)CCO3)cc(C)c1N
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1ccc2c(c1)CC(c1ccc(NC(=O)NCC(N)=O)cc1O)C2
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CC(Nc1ccc2c(c1)CCC2)C(=O)Nc1ccc(C(N)=O)cc1O
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1cc(C=CC(=NCCO)C2CC2)c2[nH]c(=O)c(C(N)=O)cc2c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CC=Cc1cc2[nH]cc(C(=O)NC3=CCCOC3)c2cc1CC(N)=O
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CCNC(=O)NC(N)c1cccc(Oc2ccc(C#CCO)cc2)c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1ccc2ccc(NC(=O)NC(=CC(=O)NC3CC3)CO)cc2c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N C#Cc1ccc(CNC(=O)NC(=Cc2ccccc2O)C(N)=O)cc1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CC(=CC=C(Oc1ccc2ccccc2c1)C(N)=O)CCC(=O)NN
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1ccc(CN(CC2=CC(O)OC=C2)C(=O)c2ccc[nH]2)c(N)c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1ccc(C=CC(=O)NNC(=O)NCc2cc(C)ccc2O)cc1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N NCc1ccc(C(=O)c2ccc(C(C=O)=CCNC(N)=O)cc2)cc1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N C=c1oc2cc(NC(=C(NC(N)=O)C(C)=O)C3CC3)ccc2c1=CC
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CC(=O)NNC(=O)C1(Nc2cc3cc(C)c(C)c(C)c3cc2O)CC1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N C#CCNC(=O)Nc1cc(OCC#C)ccc1C=Cc1c[nH]cc1O
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1ccc(C(=O)NNC(=O)NCC=Cc2ccc(O)cc2)c(C)c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N C=C(C(N)=O)c1ccc(C)c(NC(=O)NCC(O)c2ccccc2)c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1ccc(NNC(=O)c2ccc3c(c2O)C(CO)CC(N)C3)cc1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N NC(=O)c1cccc(NCc2ccc(OC3CCNC3)c(CO)c2)c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1ccc(C)c(CC(=O)NNC(=O)NCc2ccc(CO)cc2)c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CCC(=O)NC(C(=O)NNc1cccc2cc(O)ccc12)C(C)(C)C
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CC(=CN)Cc1ccc2c(c1)CCN2C(=O)Nc1ccc(O)c(O)c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N O=C(NN=C(C1=CCNC=C1)c1cccc(O)c1)c1ccccc1O
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CC(C)=CC(=O)NNC(=O)NCC(O)c1ccc2cc(C)ccc2c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N C#Cc1cccc(NC(=O)c2ccc(C)c(NC(=O)NCCO)c2)c1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Cc1cc(C2CC2)ccc1C(=O)Nc1ccc(C(N)=O)cc1C(N)=O
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N O=CNC(=O)NCC(Nc1ccc(O)cc1)c1ccc2c(c1)CCC2
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CCc1ccc(NC(=O)C(=Cc2ccc(C)c(O)c2)NC(N)=O)cc1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N CNC1C=C(c2cc(C(N)=O)[nH]c(=O)c2-c2ccc(C)cc2)C=CO1
c1ccc2c(c1)C(=O)c1c(C2=O)c(cc(c1N)C(=O)NCCCC)N Nc1ccc(NC(=O)Cc2ccccc2)cc1NC(=O)C1CCC1O
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CCOCc1cc2cc(Nc3nc4n(n3)C=CCS4)ccc2o1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C N#CCCN(Cc1nc(S)co1)C(=O)c1cc2ccccc2[nH]1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C COC(=O)C1CSc2nnc(Nc3ccc4ccccc4c3)n21
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CCSc1nc2ccc(OC)c3c4c([nH]c(n1)c23)N=C(C)OC4
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CC=Nc1nc2cc(NC(=O)c3noc4c3CCC4)ccc2s1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CCOc1ccc(NC=NC(=O)Cc2csc3nccn23)cc1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C COC(=O)c1ccn(Cc2n[nH]c(=S)n2-c2ccc(C)cc2)c1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C Cc1[nH]c(-c2nc(-c3cc4c(s3)COC4)no2)c2c1CCN2C
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C Cc1cc(C(=O)Nc2ccc3c(c2)OCN3C)c2cnsc2n1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C O=C(C=Cc1cn2c(C3CCCC3)nnc2s1)Nc1ccoc1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CN(Cc1ncc(C=O)s1)C(=O)Nc1ccc2c(ccn2C)c1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CCc1nn(C)c2c1CC(C(=O)Nc1cccc3oncc13)S2
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CN(Cc1ccsc1)C(=O)Nc1cnc2oc(C3CC3)nc2c1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C COC(=O)N=c1[nH]c(-c2ccccc2)nn1-c1ccc(S)cc1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CC=Nc1ccc(O)cc1NC(=O)C=Cc1cn2ccsc2n1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C COC(=O)CSc1ncnn1-c1ccc(-c2cc[nH]c2)cc1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C Cc1nnc(SCC(=O)N=c2ccc3c(C)cccc3[nH]2)o1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C O=C(C=Cc1cc(=O)n(-c2ccncc2)c(=S)[nH]1)c1ccc[nH]1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C Cc1cncc(-c2ccc(NC(=O)CSc3nnco3)cc2)c1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C COc1cccc2[nH]c(-n3c(CN4CCCC4)csc3=O)nc12
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CC=C(C)OCc1ccn2c(=NC(=O)c3cccs3)[nH]nc2c1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C O=C(OCC=Cc1cn[nH]c1)c1cnc(Nc2ccccc2)s1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C Cc1ncc(COc2cccc(NC(=O)c3cnccn3)c2)s1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CCOC(=O)c1cncc(Nc2ccc3cnn(CS)c3c2)c1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C O=C(Nn1ccnc1)c1ccc(Cc2nc3c(o2)CSC3)cc1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C N#Cc1c[nH]c(=O)c(CSCCOc2ccc3cccn3n2)c1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CC(=O)C=Cc1ccn(-c2cc(N=C(C)c3cncs3)no2)c1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CCc1nc2cc(NC(=O)c3cnc(SC)nc3C)ccc2o1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C CCC(=O)Nc1csc2c1nnn2C(=O)c1ccc(CC)cc1
N(C(=O)C1CC1)c1sc(c(c2ccccc2)n1)c1nc(no1)C Cc1cc2c(nn1)Cc1sc(C(=O)NN=Cc3ccco3)cc1-2
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1ccc(OC(=O)N=c2[nH]c3ccc(OC)cc3s2)cc1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC CC(=O)OCC(=O)Nc1cccc(Sc2nc3ccccc3o2)c1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC CSCc1oncc1C(=O)Nc1c(C)cc2coc(=O)cc2c1C
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COC(=O)c1ccc(Oc2cc3cc(C(C)C)sc3[nH]c2=O)nc1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC CC(=O)Oc1cscc1C(=O)Nc1ccc2oc(C3CC3)nc2c1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1cc2c(cc1C(=O)N=c1[nH]c3ccc(C)cc3s1)OCO2
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1ccc2c(ccc3csc(N=CCC(=O)NC(=O)O)c32)c1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC CCOC(=O)c1cc(CSc2nc3ccccc3c(=O)[nH]2)oc1C
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1ccc(OCCN=c2[nH]c3ccccc3s2)cc1OC
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC CCc1ncc(C=CC(=O)NCc2c(C)oc3cscc3c2=O)o1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC CCOCc1ccc(-c2csc(=NC(=O)C=Cc3ccco3)[nH]2)o1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1cccc(NS(=O)(=O)c2cc3ccccc3n2C(C)=O)c1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC OCCc1cnc(-c2ccc(Oc3ccc4c(c3)OCO4)nc2)s1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1ccccc1OC(=O)C(=Cc1ccoc1)Sc1ncc[nH]1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1ccc(NC(=O)C=Cc2cccs2)cc1Oc1cnoc1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC Cc1nc(C=Cc2ncc(C=CC(=O)c3occ(C)c3O)o2)cs1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC Cc1sc(Nc2ccc3c(c2)OCO3)nc1COCc1ccco1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COCc1ccc(C=CS(=O)(=O)Nc2cccc3oncc23)cc1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC C=NC(=O)c1ccc(O)cc1C(=O)OCc1nc2ccccc2s1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1ccc2sc(=NC(=O)c3ccc(OC)c(OC)c3)[nH]c2c1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC Cc1cc(OCc2ncc(C(=O)Oc3cccc(O)c3)s2)ccn1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1ccc2c(SCC=O)c(-c3cc(C)oc3OC)[nH]c2n1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC C=NC(=O)c1cc(CNC(=O)c2cc3cccc(OC)c3o2)cs1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC Cc1oncc1C(=O)OCc1ccc(O)c(N=Cc2cccs2)c1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC O=C(C=Cc1cc(O)c2c(c1)OCO2)N=c1[nH]c2ccccc2s1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COC(=O)c1csc(-c2cccc(Oc3cccc(O)c3C)n2)n1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COCC(=O)Nc1ccc(C(=O)Oc2ccc3ccsc3c2)nc1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC Cc1nc2c(cc1NC(=O)CCCS(C)(=O)=O)oc1ccccc12
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1ccc2onc(OCC(=O)Nc3ccccc3SC)c2c1
c1ccc(cc1)c1c(sc(n1)NC(=O)c1ccco1)C(=O)OCC COc1ccc(-c2nc(C=CC(=O)O)c3ccsc3n2)cc1OC
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COCc1cc(C)cc(-n2ncc(C(=O)OCCOCc3ccncc3)n2)c1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COC(=O)COc1ccc2cnc(C(=O)N(C)Cc3cc(C)nn3C)cc2c1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CCN(CCc1nc2c(C)ccc(OC)c2o1)C(=O)Cn1nc(C)ccc1=O
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC C#CCOC(=O)c1c(C)c(C(=O)Cn2cccc2)c(C)n1Cc1nc(C)no1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COc1coc(COc2ccc(-n3c(C)nn(C)c3=NC(=O)C(C)C)cc2)c1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CN(C)C(=O)Cc1ccc(C(=O)Cc2ccc(OCc3nncn3C)cc2)o1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC C=CC(=CC)OCCOc1ncccc1Oc1cn2c(C)cnc2n(C)c1=O
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COc1ccc(OCC(=O)N(C)c2cc(-n3ccc(C)c3)ncn2)cc1OC
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CCn1cc(C(=O)c2cc(C)ccc2C)n(C(=O)Cn2ccc(OC)n2)c1=O
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COc1ccc(C=CC(=O)c2cc3[nH]ncn3c2C)c(OCC(=O)N(C)C)c1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CCn1c(CN(C)C(=O)COC(=O)C=Cc2ncc(C)o2)cc2cnccc21
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COc1ccc(OC(C)=Cc2cccn(Cc3nncn3C)c2=O)cc1OC
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COCCOC(=O)c1ccc2nc(-c3nccn3CC(C)C)c(=O)n(C)c2c1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CCc1ccc(CC(C)N(C)C(=O)c2cnc3c(c2)c(C(=O)OC)nn3C)o1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CCCOc1ccc(Cn2c(=O)n(C)n(C)c2=O)cc1Oc1cccc(C)n1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COC(=O)C(c1cn(-c2ccccc2)nn1)N(CCC1CO1)Cc1ccco1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CCCCOc1ccc(-n2nc(COC(=O)c3cnn(C)c3)cc2C=O)cc1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COC(=O)COc1ccccc1CN(C)c1noc(CCc2ccncc2)n1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COCCN(C)C(=O)c1cc(-c2nc3ccccc3o2)c(N(C)C(C)=O)n1C
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC Cc1nncn1Cc1ncc(CC(C)C(=O)COc2cccc3c2OCC3)o1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC COCC(C)Oc1cccc(-n2ncn(CCOc3ccc(C)cc3)c2=O)n1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CCn1c(C)c(C(=O)N(C)Cc2ncc(-c3ccc(OC)cc3)o2)n(C)c1=O
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CCN(C(=O)c1ccc(OC)cc1OC)C(C)c1nc(=COC)c2nccn12
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CC(=O)N(C)c1ccc(OCCOC(=O)Cn2c(C)cc3cncnc32)cc1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC Cc1cn(C)c(=NC(=O)COc2ccccc2OC(=O)c2ccn(C)c2)n1C
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC C=CCN(C)C(=O)Cc1onc2c1cnc(=O)n2C=Cc1oc(C)cc1C
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CCc1ccc(COC(=O)C(C)OC(=O)C(C)c2nc3ncccn3n2)cc1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CC=c1cnn2c(=NC(=O)CCOc3ccc(OC)cc3OC)cc(C)nc12
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC Cc1cc(C)n2c(C(=O)N(Cc3ccc(C)o3)CC3COCCO3)cnc2n1
n1(c(=O)n(CC)c2c(c1=O)n(c(n2)/C=C/c1cc(c(cc1)OC)OC)C)CC CN(Cc1c[nH]nn1)C(=O)COc1ccccc1OCCOc1ccccc1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1c(CCO)nc(N=C(N)Nc2ccc3c(c2)cc(C(=O)Nc2cc(C(C)O)ccc2C(=O)N(C)C)n3C)c2ccnn12
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1ccc2c(=NNC(=O)CCCN(CC(=O)Nc3ccc(N)cc3)C(=O)c3ccc4n[nH]cc4c3)c(O)n[nH]c2c1C
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O COCCNC(=O)C(C)Cn1cc(C(=O)NCc2cnc(-c3c(C)[nH]c4cnc(N)cc34)nc2)cc(-c2ccncc2)c1=O
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1ccc(-n2c(CC(N)C(=O)O)nnc2-c2ccc(C)c(NC(=O)c3ccc(C=CC(=O)N=c4[nH]cn[nH]4)cc3)c2)cc1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1cc(CN(CC(O)CO)c2nccc(=O)n2C(=Nc2c(C)cccc2-c2cc(N)[nH]n2)Nc2ccncc2)ccc1O
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCNCC1CNC(=O)CC1OCCc1ncc(C=NNc2c(C)c3cc4c(=O)[nH]c(=O)[nH]c4nc3c3ccccc23)cn1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O C=c1occ(C=NNC(=O)c2nn[nH]c2CCCCc2cccc(-c3n[nH]c(NC(=O)C=Cc4ccc(O)cc4)n3)c2)c1=C
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O COc1cc2c3c([nH]c2cc1OCCN)CN(C(=O)NCCc1n[nH]c(C(C#N)=Cc2ccc4ccc(=O)[nH]c4c2)n1)CC3
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCNC(=O)c1c(C)cc(OCC=Cc2coc3nc(N)c(-c4nc(CCc5ccc(NN)nc5)nc(=O)[nH]4)cc23)cc1C
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O C=CCNCc1ccnc(NC(=O)c2nc(-c3cn[nH]c3COc3cc(C(N)=O)cc(-c4ccc(OCC)cc4)c3)n[nH]2)c1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCc1nccn1-c1cncc(NC(=O)C(=Cc2cccc(C(N)=O)c2)NC(=O)Cc2cc(C)nn2-c2ccc(O)cc2)n1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC(C)c1cccn1-c1cc(NC(=O)CC(CNC=O)C(=O)NNc2cccc(Oc3ccc4cncnc4c3)c2)[nH]n1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O NC(=O)CCN(CCC(=O)N1C=CCC1C(=O)Nc1cccc2[nH]ccc12)C(=O)C=Cc1nnc2c3ccccc3[nH]n12
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCc1nc(NC(=O)c2n[nH]c(C)c2C(=O)Nc2ccc(C)c(C(=O)c3ccc(C)cc3)c2)nc(-c2c[nH]c(C(N)=O)c2)n1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O COc1ccc(Nc2nc(N)c3cn(-c4ccccc4OC(C(N)=O)C(=O)NCCc4ccc(C#N)cc4)nc3n2)cc1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1ccc(CNC(=O)C(=O)NNC(=O)CN(C)C(=O)c2ccccc2)c2c1ccn2-c1ccc2nc(CCNN)[nH]c2c1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O COc1cccc(NC(=Nc2nc(-c3c(C)n(Cc4ncco4)c4ccccc34)[nH]c(=O)c2N)NC(C)C(=O)NC2CC2)c1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1c(NC(=O)NCc2cn3cc(C(=O)Nc4cncnc4)ccc3n2)ccc(-c2ccncc2)c1C(=O)NC(C)(C)CO
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCCNc1c(NCCNc2nc(=O)c3cnc(NC(=O)c4cccc(C=Cc5coc(=O)[nH]5)c4)nc3[nH]2)ccc(C)c1C
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1ccc(NC(=O)CCNc2nc(N)nc3ncc(C=NNC(=O)C=Cc4cn(C)c5cccc(O)c45)c(C)c23)c(O)c1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O C=Cn1nc(C(C)(C)N)c(CCc2c(N)n(-c3cccc(C(=O)Nc4ccc5ccn(C)c5c4)c3OC)c(=O)[nH]c2=O)c1N
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1ccc2[nH]c(=O)n(CC(=O)Nc3ccc4cc(NC(=O)C(=O)NCCCc5cccc(NN=CN)n5)ccc4c3)c2c1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CNC=CC(=O)Nc1ccc2oc(-c3c(NC)nc(N)c(C(=O)N(Cc4cn[nH]c4)Cc4ccc(C5CC5)o4)c3C)nc2c1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1cc(C(=O)NCCc2cn(CC(NC(=O)N(C)CCO)c3ccccc3C(=O)c3cnn[nH]3)c3ccccc23)ncn1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1ccc(C)c(OCc2c(-c3cc(N(CC(=O)NCCC(C)O)Cc4cn[nH]c4C)c4c(c3)[nH]c(=O)n4C)n[nH]c2N)c1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC(C)(O)Cc1ccc(-n2ncc(-c3ncc(C(=O)NOc4ccc(Nc5ccc(OCCC#N)cc5)nc4)[nH]3)c2N)cc1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O COCc1cc(NC(=O)NCc2ccc(-n3cnc(C(=O)NN=Cc4ccc(-n5ccnc5C)cc4)n3)cc2)cc(O)c1C
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O COC(N)CNC(=O)OC(C)C=c1c2c(N)nc(Oc3ccc(C)c(CN4CCN(CC#N)CC4)c3)nc2n2c(C)ccc12
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1ccc(Nc2ccnc(NC(CO)C(=O)Nc3ccc4cccc(C(=O)Nc5cnn(CC(O)CN)c5)c4c3)n2)cc1
n1(c2c(nc1)c(nc(n2)NCCc1nc[nH]c1)NCC(c1ccccc1)c1ccccc1)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCN(C)C(=O)c1cc(NC(=O)c2[nH]c(C)c3c4c([nH]c23)CN(CC(=O)Nc2cccc3nnc(O)cc23)CCC4)ccn1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CCc1ccc(C[NH+]2CCNCC2C(=O)Nc2ccc3nc4c(cnc5nnnn54)cc3c2)o1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N C=[NH+]c1ncnn1-c1cc(Nc2ccc3cnn(-c4ccccc4)c3n2)cc(=O)n1CCOC
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N Cc1ccn2c(Cn3c(NC(=O)C=Cc4ccc([NH3+])cc4)nc4c(cnn4C)c3=O)nnc2c1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N C[NH+](CC#N)Cc1ccc(-c2nc3[nH]c(=O)c(=Cc4ccc(Nc5ccncc5)nc4)n3n2)o1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N COc1c2c(=O)[nH]c3[nH]n(C)c(=Nc4ccc(-c5ccnn5CC[NH+](C)C)cc4)c3c2nn1C
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CNC(=O)c1ccc(C=NN(Cc2ccncc2)c2nn3c(=O)cccc3n3nc[nH+]c23)cc1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N Cn1cc(CN2Cc3[nH+]c4c(nnn4-c4ccc(C(N)=O)cc4)n3-c3ccccc32)nc1CO
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CNc1nn2c3ncnc(Oc4ccccc4OCc4ccccn4)c3nc2n1C1CC[NH2+]C1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N C[NH+](C)CC(Nc1n[nH]c(-c2cncc(OCc3nc4ccccc4o3)c2)n1)c1ccncn1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N Cc1ccc(C[NH+](C)c2ccc(C(=O)N=c3[nH]nc4n3ccc3nc(C5CC5)nn34)cc2)o1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N Cn1nccc1C(Oc1ccc([NH3+])cc1)c1ncccc1CC(=O)Nc1cncn2cnnc12
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N Cc1ccc(-c2nnc(-c3ccc4c(c3)nc3[nH]cnn34)o2)cc1C(=O)N1CCN(C[NH3+])CC1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CC[NH2+]Cc1ncnn1-c1nn(C)c2ccc(Cn3c(-c4ccc(OC)cc4)n[nH]c3=O)cc12
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N C=C1C[NH+](Cc2nc(Cc3ccc(-n4ccc(C)n4)cc3)cc(=O)[nH]2)C(c2nnno2)CC1=N
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CNC(NCC(=O)n1c(C)c2c3c1cnn3ccn2N=CC=N)=[N+](C=O)Cc1ccc(C)cc1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N COC(=O)CCc1nc2nc(Nc3ccc(Cc4n5cc[nH]c5c(C)[n+]4C)cc3C)nnc2[nH]1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N C[NH2+]CN1N=CC=NC1=Cc1n[nH]c(=NC(=O)c2cccc(Cc3nc4ccccc4o3)c2)[nH]1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N C=C1c2cc(CNC(=O)c3cncc(NCc4nc5nc(C)ccn5n4)[nH+]3)ccc2OCN1C
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CC1=CC(n2nc(-c3ccco3)nc2N=c2c3cc4ccn(C)c4nc3n(C)n2C)C[NH2+]CO1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N Cc1cccc(CNC(=O)C=Cc2ccc(-n3nnnc3N=Cc3cnc4c(n3)C[NH2+]C4)o2)c1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CNc1nnc(NCc2ccc(Oc3ccc(-n4cncn4)cc3)c(C=O)c2)c2[nH+]c(C)cn12
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CC(=O)c1ccc(C=Cc2nnnn2-c2ccc(C(=O)N=c3[nH]cnn3C(C)=C[NH3+])cc2)cc1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N C=CCN(Cn1nc(C)c2cc(C(=O)N=c3[nH]nc4ccccn34)c[nH+]c21)C1COCC1C
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N C=C(C[NH+](C)c1ccc(CCc2ccc(C(=O)N=c3[nH]nn[nH]3)cc2-n2ccnn2)cc1)OC
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N Cc1cc2c(cc1Oc1ccc(Nc3nncc(N4CC(=O)n5ccnc5C4)n3)cn1)C[NH+]=C2
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N Cc1nc2c3c(ccn2c1C(=O)Nc1nc2c(c(C)nn2C)c(=O)[nH]1)N(C(C)C)CC[NH+](C)C3
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N COCC[NH2+]c1cc(=O)n(-c2ccc(Nc3ncnc4c3Cc3ccccc3N4C)nn2)cn1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CC=CC(=O)c1c(C)cc2nnc(N=C(N=c3nc(C)oc(=[NH2+])[nH]3)Nc3ccccc3)n2c1C
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N CC[NH+]=C(OC1CC1)c1c[nH]c(=NC(=O)Cc2cc(-c3cnc(-n4cccc4)nc3)nn2C)[nH]1
n1c(n2c(nc(n2)c2ccco2)c2c1n(cn2)CC[NH+]1CCN(CC1)c1ccc(cc1)OC)N C(=NNc1cc(N2CCOCC2)n2cc(-c3ccc(Oc4cccnc4)cc3)nc2n1)C1=[NH+]N1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1c[nH]c(C(=O)O)c1CCN(CC(N)=O)C(=O)NCC(=O)NNn1cccc1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1[nH]nc(N2CC(CO)OC(CO)C2)c1NC(=O)C(=O)Nc1ccc(N)nc1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1cc(CCNC(=O)CNC(=O)NNC(=O)c2ccc(NC=O)c(O)c2)[nH]n1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCOc1cc2c(cc1OC)c(C(=O)N=CN)cn2N=C(N)C(=O)NCC(N)=O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1nc(=O)cc(C=NNC(=O)NCc2ccc(OCC(N)=O)c(C(N)=O)c2)[nH]1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O NNC1COc2c(NC(=O)CNc3ncncc3N)ccc(OCC=O)c2OC1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O O=C(NCc1n[nH]c(=O)[nH]1)Nc1ccc(NC(=O)C2CC(=O)N(CCO)C2)cc1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC(O)c1[nH]c(=O)c(C(=C(N)N)c2nc(C3CN(C)CCO3)no2)cc1C(N)=O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1cc(NC(=O)C(=O)Nc2c[nH]c(C(=O)NCCOCNN)c2)c(C=O)cn1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC(Cc1ccco1)(NC(=O)N=C(N)NCc1ccnc(OCCO)n1)C(N)=O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCN(C(=O)c1cn[nH]c1)c1cc(N)cc(NC(=O)NC(=O)C(=O)NCCO)c1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC(C)(Cc1cc(NC(=O)C(=O)Nc2cn[nH]c2)c(=O)[nH]c1N)C(=O)NCCO
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Nc1ccc2c(c1)C(=O)C(=O)N2CCNC(=O)Nc1nc(N)cc(OCCO)n1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1[nH]c(C(=O)NNC(=O)NN=Cc2ccoc2)cc1C(=O)CNC(=O)CCN
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CN(C)c1ccc(NC(N)=O)cc1C(=O)NCC(=O)NNC(=O)c1c[nH]cc1O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1nc(C)c(CC(=O)NCCC(=O)Nc2cc(C(N)=O)c(N)[nH]c2=O)c(=O)[nH]1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCn1c(CO)nc(O)c(C(=O)NNC(=O)NCCCc2cccc(N)n2)c1=O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCC(NC(=O)NCC(=O)N(Cc1cn[nH]c1)Cc1ccc(C(N)=O)o1)C(N)=O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O NC(=O)c1c(NC(=O)CCCC(=O)NCC=Cc2cnc(N)o2)cn[nH]c1=O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC(NC(=O)c1ccncc1C(=O)NN=Cc1ccc(CNC(N)=O)o1)C(N)=O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CNc1ncc(C(=O)NNC(=O)NCC(O)C(=O)Nc2ccccc2C)c(=O)[nH]1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O NC(=O)NNc1ccc(OCC(O)CNc2nc(N3CCC3)c[nH]c2=O)c(O)c1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O NNC(=O)C=C(C=CC(=O)Nc1ccc(OCC=O)cc1)N=C(O)c1ncn[nH]1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC(C)C(O)=C(CNC(=O)NNC(=O)c1cccc(N)n1)C(=O)n1cn[nH]c1=O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CCN(CC(=O)NNC(=O)NCc1cc(O)ccc1OC)C(=O)c1cc(N)[nH]n1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC(C=O)CN(C)C(=O)CNC(=O)n1nc(C(N)=O)c2cc(NC(N)=O)ccc21
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O Cc1ocnc1CN(CCO)CCC(=O)NNC(=O)c1cc(C#N)c(N)[nH]c1=O
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O NC(=O)C(=CO)NC(=O)CNC(=O)NCCCc1ccc(-c2n[nH]c(=O)[nH]2)cc1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC1=NC(=O)CC(NN=C(C(N)=O)C(=O)Nc2ccc3c(=O)[nH]c(=O)[nH]c3c2)=C1
n1(c2c(nc1)c(nc(n2)N[C@H]1[C@H](O)CCC1)N)[C@H]1[C@@H]([C@@H]([C@H](O1)C(=O)NCC)O)O CC(NC(=O)C(NC(=O)NCCc1nc(-c2ccccc2)no1)C(N)=O)C(N)=O
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 CCCCn1c(=O)n(-c2cccc(-c3c[nH]nc3C)c2)c(=O)n1-c1cc(F)ccc1F
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Cn1nc2ccc(C=NNC(=O)c3cccc(OCc4cc(F)ccc4F)c3)cc2n1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 CCN(Cc1cc2ccc(Oc3ccc(F)cc3F)cc2c(=O)[nH]1)Cc1nncn1C
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 CN(CCn1cccc1)C(=O)c1cc(F)ccc1NC(=O)c1cnc2ccc(F)cn12
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 C=CCN(c1ccc(C)cc1)c1nn(-c2nc3cc(F)c(F)cc3[nH]c2=O)cc1C=O
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 C=c1c(=O)[nH]c2nnc(CN(Cc3ccc(C4CC4C)o3)c3ccc(F)c(F)c3)n12
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Cc1cc(Cc2nc(-c3ccc(F)c(Oc4ccccc4F)c3)nc(=O)[nH]2)nn1C
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Cc1ccc(COc2c(F)cc(F)cc2C(=O)NN=Cc2cnn3cccnc23)cc1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Cc1ncnc2[nH]c(=NCc3ccc(C(=O)OCc4ccccc4F)c(F)c3)n(C)c12
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 O=C(Cc1ccccc1OCc1ccccc1F)N=c1[nH]nnn1-c1ccc(F)cc1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Cn1c(=NC(=O)c2cc(F)cc(OCC(F)=Cc3ccncc3)c2)[nH]c2cnccc21
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 CCc1cc(OC)c(=NC(=O)Cn2c(-c3ccc(F)c(F)c3)nc3ccccc32)[nH]n1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 COc1ccc(C=Cc2nc(-c3cc(C)c(F)[nH]c3=O)nc(-n3cccc3)n2)cc1F
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 O=C(c1ncccc1NN=Cc1cc2ccccc2n(CC(F)F)c1=O)n1cccc1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 O=C(Oc1ccc(F)cc1F)c1cccc(NCn2ccnc2Cn2ccnc2)c1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 O=C(CC=Cc1nc(-c2cccc(F)c2)no1)N=c1[nH]c2ccccc2n1CCCF
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 CC(=O)Nc1cc(-c2ccc3oc4nnc(C5CC(C)CN5C)n4c3c2)ccc1F
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 COCCCc1nc(F)c2c(=O)nc(Nc3ccccc3)n(-c3ccc(F)cc3)c2n1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Fc1ccc(F)c(Oc2ncc(C(c3nc4ccccc4o3)N3CCNCC3)cn2)c1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 CC(C)c1nc(-n2ccnc2)c2ccc(C(=O)Nc3ccc(C(F)F)cc3)cn2c1=O
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Cc1ccc(-n2ncc3c(F)cc(C(=O)NN=Cc4cccc(OCF)c4)nc32)cc1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Cc1ccc(NC(=O)c2cc(C=O)nc3cc(-c4nc(F)cn4C)n(C)c23)c(F)c1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Cn1cc(-c2cc(N3CCCCC3CF)ncc2-c2nnco2)c2cc(F)c(O)cc21
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 O=c1[nH]nc(C=Cc2ccccc2)n1N=Cc1ccc(Oc2cc(F)cc(F)c2)nc1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 O=C(Cn1ncnc1CCCF)Nc1ccc(Oc2ccc3c(F)ccnc3c2)cc1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 CNc1c[nH]c(=NC(=O)c2ccc(OCc3ccc(C)cc3)c(F)c2F)n2ccnc12
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 COC(=O)c1nc(N=c2[nH]c3cc(F)ccc3n2-c2cccc(F)c2)c(C#N)cc1C
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 Cc1ncc(-c2nc3ccc(CN(C=O)CCOc4ccc(F)c(F)c4)cc3[nH]2)cn1
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 CN(C(=O)Cc1cnc(-c2ccc(CC3CC3)o2)[nH]1)c1cc2cnn(C)c2cc1F
n1c(nc2c(c1)n(c(=O)n2c1cccc(c1)OC)Cc1c(cccc1F)F)NC1CC1 CCOc1ncc(NC(=O)C(c2ccc3ccncc3n2)c2ccc(F)cc2F)cn1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 COc1ccccc1-c1ncc2c(N)c3nnc4c(cnn4C(CCO)CCCO)n3c2n1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cc1ccc(OCCn2nc3c(c2NCc2ccncc2)c(=O)[nH]c2nc(CO)nn23)cc1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 O=C(COc1ccc(-c2noc(CNc3ccc4cn[nH]c4c3)n2)cc1)NCc1c[nH]cn1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cc1cc(OCCNc2nc3ncnn3c3[nH]c4c(C)oc(C)c4c23)cc(C)c1OCN
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cc1ncc(C(=O)Nc2cc3ccc4cc5c(cc4c3cn2)[nH]c(=O)n5CC(O)CN)nn1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cn1c2cccnc2n2c(-c3ccccc3)nc(-c3nnc(CC(=O)NC(CN)CO)o3)c12
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 NCCNC(=O)c1ccc(-c2n[nH]c3nc4cc(COc5cc[nH]c(=O)n5)ccc4n23)cc1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cc1cnn(-c2ccc(NC(=O)c3c(C)nc(Nc4cc(C)nn4CCO)[nH]c3=O)cc2)c1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 CC(=O)NNc1nncn1N=Cc1ccc(OCC(=O)Nc2cc(C)c3[nH]ccc3c2)cc1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 COc1ccc(-c2nc(O)n3nnc(CNc4ccccc4-c4cc(CN)no4)c3n2)cc1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cc1[nH]c(-c2cnn(-c3cnnc(NCCO)c3)c2C)nc1CCC(=O)NCc1ccoc1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 CCOc1c(C)cc(CC(=O)NCc2nc(-n3nc4[nH]ccc4c3N)n(C)c(=O)n2)cc1C
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 COc1ccc2cc(CNc3nc4n[nH]c(Oc5cncc(N)c5)c4c(=O)[nH]3)ccc2n1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cc1cnc2[nH]c(=NNC(=O)COc3ccc(Cc4n[nH]c(C(C)C)n4)cc3)[nH]c(=O)c2c1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 C=C(N)CNC(=O)c1cc(-c2cc(-c3cn[nH]c3)nn2C)nn(Cc2ccc(CC)o2)c1=O
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 CNCCNc1ccc(NC(=O)C(=O)Nc2cccc(-n3cc4c(O)nn(C)c4n3)c2)cc1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 CCN=CCNC(=O)NCCc1[nH]c2c(C(=O)Nc3ccc4onnc4c3)cncc2c1C
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cn1c(=O)n2c(O)c(N3CCC(CO)C3)c3c(CNc4ncnc5cnccc45)cnc1c32
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 CC=CC(=Cc1cnn(C)c1)OC(C)C(=O)NNC(=O)c1c[nH]c2c(-c3cc[nH]c3)n[nH]c12
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 O=C(Nc1ccccc1NCc1c[nH]cn1)c1nc2[nH]c(=O)c(=Cc3cccc(O)c3)n2n1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 CCc1c(C)nc(-n2nn[nH]c2=NC(=O)c2ccc(C=CC(=O)OC)cc2)c2cc(N)[nH]c12
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cn1c(COc2ccc3ccc(N)nc3n2)nnc1-c1cc(C#N)c(O)cc1OCCCN
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 CCCN(c1nc(=O)n(CNC(=CNC=O)c2cc(C)n(C)c2)[nH]1)c1nc2ccccc2o1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 C=c1nc(-n2nnnc2CNC(=O)Nc2ccc(Oc3ccccc3OC)cc2)[nH]c1=CC
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Cc1oc(-n2ncn3[nH]c(=O)nc23)c(CC(=O)NCc2cc(C)n(C3=CCN=C3)c2C)c1C
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 CC(=O)c1ccc(N(c2ccc(O)c(C=O)c2)c2nc(NN=c3cc(C)[nH]cn3)n[nH]2)cc1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 COc1cccc(NC(=O)CC(=O)N=c2[nH]nc(NCc3nn(C)c4cc(C)ccc34)[nH]2)c1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 C=C(CN)Cc1nc(-c2ccccc2-n2c(C)nnc2OCCC(=O)Nc2cc[nH]c2)no1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 COc1ccc(NC(=O)C=C(C)N=c2[nH]nc3c4c(ccn23)oc2c(C)c(=N)[nH]nc24)cc1
n12c(c3c(nc2N)n(nc3)CCc2ccc(N(CCO)CCO)cc2)nc(n1)c1occc1 Nc1nn2cccnc2c1NC(=O)c1ncc2ccc(COc3ccc(CO)cc3)nc2n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CC=c1cc(NC(=O)Nc2ccc(-n3cnnc3Cn3nnnc3C)cc2)ccc1=C(F)F
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CN=c1ccc(-c2nn(-c3ccc(F)cc3)cc2CNC(=O)C=Cc2nnc(F)n2C)n[nH]1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cc1nc(NCc2cccnc2N2CCNC2C(=O)F)nn1-c1nn(C)c2cc(F)ccc12
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CN(C)CCn1cc(F)cc(N=c2[nH]nncc2Nn2ccnc2-c2ccccc2F)c1=O
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CN(C=N)c1ccc(C(NC(=O)c2cnnn2C)c2ccc(F)c(-n3cncn3)c2)cc1F
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cc1nc2n(C3=C(Nc4ccccc4)C(=O)N(C)C(CF)N3)nc(-c3cncc(F)c3)n2n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CC1COCc2ncc(CNc3ccc(NCc4nnc5cnc(C#N)cn45)c(F)c3)n21
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CNc1cn(C)c2nc(-c3ccc(N=C(N=C4NCCN4CF)c4ccc(F)cn4)o3)cn12
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CNc1nc(=C2C(F)=C(NC(=O)CCc3ccc(F)cn3)C(C)n3ccnc32)n2cnnc12
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cc1cc(-n2nccc2NCC(F)F)nc(Nc2ccc(-n3c(C)nncc3=O)cc2)n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CCc1nn2c(-n3ccnc3C)n[nH]c2c1CNC(=O)N1CCc2cc(C(F)F)ncc2C1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C O=c1[nH]cncc1-n1nnnc1C=Cc1ccc(Cc2nc3c([nH]2)CCCN3C(F)F)cc1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C N#CCCN(Cc1nc[nH]n1)c1ccc(CNC(=O)Cn2nnc3cc(F)ccc32)cc1F
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CNC(=N)c1n[nH]c(-c2cnn(-c3ccc(F)cc3F)c2-n2c(C3CC3)nc(C)cc2=O)n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cc1nnc(Nc2ccc3c(CN4CCCCC4)nc(=O)[nH]c3c2)n1-c1cnn(C(F)F)c1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CNCc1nn2c(CN3CCN(C(=O)Nc4ccc5c(F)cccc5c4F)CC3)nnc2[nH]1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C C=CCN(c1ncnc2c1ccc1nc(CNC(=O)Nc3cn(C)cc3C#N)cn12)C(F)F
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C O=c1[nH]c(=NCCCc2ccc(N3CCN=N3)cc2)[nH]c2c1nnn2-c1ccc(F)c(F)c1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cc1ncc(NCn2nc(-c3ncnn3-c3ccccc3)cc2C(F)F)c(C2CNOC2)n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cc1nc2nc3[nH]c(C(C)Cc4ccc5c(c4)CNCO5)nc(=N)c3c(N=CC(F)F)n2n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cc1c(CNc2cc(C(=O)NN=Cc3ccc(F)cc3F)ccn2)cnn1-c1ncn(C)n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cc1ccn(-c2ccc(-n3nc(C(F)F)cc3NCC(=O)NN=Cc3cnn(C)c3)cn2)c1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CN(C)CC(Nc1c2cnc3c(-c4cc(F)cc(F)n4)nnn3c2nn1C)C1=CCOC=C1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cn1cc(C=Nc2ccnn2-c2ccn[nH]2)c(CNCC(=O)NCc2ccc(F)cc2F)n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C O=C(N=c1cccc[nH]1)c1nc(Nc2ccn(CC(F)F)n2)n(CCCc2ccccn2)n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C O=C(CCNc1cnn(-c2cc(F)c3c(c2)ncn3N=CCF)c1)NN=Cc1cccnc1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C Cc1cc(N(C)Cc2cn3ccc(C(F)F)cc3n2)nc(=O)n1C1=NC=Cn2ccnc2N1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C O=C(Cn1cnnc1)Nc1cc(F)ccc1-n1ncc(NC=CN=Cc2ccccc2F)n1
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C CN1CC(CNc2cc(-n3ncc4cnn(C)c43)nc(C3CC3)n2)Oc2c(F)cnc(F)c21
n1c(cc2n(c1N)nc(n2)c1ocnc1)N(CCN1CCN(CC1)c1ccc(cc1F)F)C N#Cc1ccc(C=Cn2c(CNC(=O)NCc3cn4ccncc4n3)nnc2C(F)F)cc1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCc1cc(C)n(-c2cc(C)c(CC(=O)OCC3CCC(c4n[nH]c(C)n4)O3)c(C)n2)n1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCOc1cc(CC)c(C)cc1NC(=O)c1cc(CN2CCN(c3cnn(C)c3)C2)on1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CC(=CCCC#N)OCc1ccc(C(O)C(=O)N(C)c2cnc(-n3cccn3)nc2)cc1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCN(C)C(=O)C=Cc1coc(C=Cc2cnn(-c3cc(C)c(C(=O)NC)cn3)c2C)n1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C C=C(CN(CCN(Cc1cn[nH]c1)C(=O)c1nc(C)n2c(C)coc12)C1CCCC1)OC
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CN(CC=N)Cn1nnnc1COC(=O)C=C(CC(=O)c1ccccc1)c1ccccc1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCc1nccn1-c1nn2c(c1NC(=O)CCCOc1ccccc1OC)N(C)CCC2
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CC(CN1CCCC1=O)c1noc(C(C)Nc2cccnc2OCCc2ccncc2)n1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCC(=O)Nc1ccn(C(=O)CCCC(C)n2cncn2)c1COc1cccc2c1=NC=2
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C Cc1ccc(OCCN=C(N(C)CCOc2ccoc2)N2CCCC2)cc1-c1nc[nH]n1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C COC(CC#N)COCc1cc2c(C)nc(-n3nc4c(c3C)CCCCC4)nc2[nH]c1=O
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CC=Nn1cnnc1CN(C)C(=O)C(=O)Nc1ccc(C)c(-c2cc(OC)ccc2C)c1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCCCC1NC(=O)N(CCC(=O)N(C)c2ccc3c(ccn3-c3cnn(C)c3)c2)C1=O
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C COC(C)Cn1cc(C(=O)C=Cc2cnc(NC(=O)C=Cc3cccnc3)nc2C)cn1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C COc1ccccc1C1=NN=C(C(=O)Nc2cccc(COCc3nncn3C)c2C)C1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C C=CCN(CC)C(=NC(=O)Cn1cc(C#N)c2cccnc21)NCc1ccc(COC)o1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CC=CC(=O)C=C(C)C=C(C)c1cncn(CC(=O)Nc2cccn3c(C)nnc23)c1=O
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCc1cc(CN(C)C(=O)C(=O)NN=C(C)c2ncc(-c3ccc(C)cc3)o2)n(CC)n1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C COc1ccc(Oc2nc(N=C(C)NCc3nccn(CC(C)C)c3=O)ncc2C)cc1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCCN(C)CCC(=O)Nc1cccnc1-c1nnc(C(C)N2CCc3occc3C2)o1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C C=CC(C=Cc1n[nH]c(=NC(=O)COc2ccc(-c3nc(C=CC)no3)cc2)n1C)=CC
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCN(c1ccncc1)c1nccc(C(=O)NCC(=O)Oc2cc(N(C)C)ccc2C)n1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C C=CCOC(=CC=CCn1nnc(C(=O)NCc2cn(C)nc2C)c1C)c1ccc(C)o1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCCNc1nc(C(C)OC(=O)CCCc2ccc3c(c2)OCC3)nn1-c1cnn(C)c1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C COc1ccc(OC(C)C(=O)NCCCc2nnnn2-c2cc3c(cn2)CCC3)c(C)c1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C Cc1ccc(NCCn2cc(OC(=O)CCC(=O)N=c3ncccn3C)c(C)n2)cc1C
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCN(C)c1noc(-c2cc(NC(=O)C=Cc3ccc(N(C)C=O)cc3)c(C)c(C)n2)n1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCCn1cc(-c2nc(-c3nc(CN4CC(C5CC5)OCC4C)cc(=O)[nH]3)oc2C)cn1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C C=CCN(Cc1ccncn1)C(=O)c1cccc(NC(=O)c2cncnc2OCCC)c1
c1c(nc2c(c1)nc(n2CCCOC)NC(=O)c1cccc(c1)C#N)C(=O)N(C(C)C)C CCOC(C)c1nc2c(c(NCC=C(c3cccnn3)c3conc3OC)n1)CCCC2
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 Cc1cnc(CNC(=O)c2cnn(C(=O)CCC(=O)Nc3ccc4c(C)c[nH]c4c3)c2C)o1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COCc1cc(CNc2nc3[nH]ncc3cc2C(=O)OCc2c[nH]c(C(C)(C)C)n2)oc1C
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COC(=O)C=Cc1ccc(CNC(=O)C(C)Nc2ccc3c(c2)nc2[nH]nc(C4CC4)n23)o1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COC(=O)C(=CC=Cc1ccc(-c2nnn[nH]2)cc1O)Oc1nc(-c2ccc(C)cc2)c[nH]1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CCc1noc(CNC(=O)c2ccc3oc(C(=O)NCc4nc(C5CC5)[nH]c4C)cc3c2)n1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COc1ccc(Oc2ccc(-c3cnn4cccnc34)cc2NC(=O)NCN(C)C)cc1O
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COC(O)C(C)NC(=O)Oc1cc2cc[nH]c2cc1-c1nnc(N=Cc2ccc(C)cc2)[nH]1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COc1cccc(NC(=O)C(=O)NCc2cc(C)nc(Nc3ccc4oc(C)nc4c3)n2)c1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CC(=O)Cc1cc(NC(=O)c2ccccc2Nc2cn3nc(C)cc3nn2)cc(C=O)c1O
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CC(=Nc1nccn1CC(=O)NCc1coc(NC2CC2)n1)c1ccc2oc(CO)cc2c1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 Cc1cccc(Oc2cccc(C(=O)NCCC(=O)Nc3c(C)nn4ccnnc34)c2O)c1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CCCC(=O)C=Cc1c(-c2cc(-c3ncnc(Nc4cccc(OC)c4)n3)c[nH]2)o[nH]c1=O
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COC(=Nc1nc(N2CCC(OC)C2)cc2nc3ncccc3cc12)c1c(N)oc(C)c1O
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COc1ccc(Oc2cccc(C(=O)NC(C)c3nc[nH]n3)c2)cc1OCc1ncc[nH]1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CCc1ccc(C=NC(=O)c2ccc(NC(=O)NCCc3cc(-c4cn[nH]c4)no3)cc2)o1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COc1ccc(C=Cc2nc(C)cc(=O)[nH]2)cc1NC(=O)c1cn2ccc(C(C)O)nc2n1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CCNC(=O)Nc1ncccc1-c1nc(C(=O)OCCCc2ccc3cc(C)oc3c2)n[nH]1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CC(C)(C)OCCCOCc1nc2cccnc2n1Cc1nc2ccc(NC(N)=O)cc2o1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CCNc1nc2ccc(NC(=O)c3ccc(-n4cc(CO)cn4)nc3)cc2cc1C(=O)OC
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COCNC(=O)C(=O)Nc1cccc(C=Cc2nnc(Nc3ccc4ccccc4c3)o2)n1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 Cc1cn(-c2ccc(OCc3cnc(N)c(C#N)c3)cc2Oc2cc(CO)ccn2)c(=O)[nH]1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CCC(=N)COc1cc2cc(C)oc2cc1C=CC(=O)NNC(=O)c1n[nH]c2ncccc12
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 COc1cc2c(cc1OCCN)[nH]c1nc(C)nc(NC(=O)c3onc4c3CC(C)CC4)c12
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CCC(NC(=O)c1coc2ncnc(ONC(=O)CCc3ccccc3)c12)c1ncc(C)[nH]1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CN(C)C(=O)c1ccc(Nc2nc3cc(NC(=O)Cc4noc5c4OCC5)ccc3[nH]2)cc1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 Cc1[nH]cc(C(=O)Nc2ccc3c(c2)nc(C2CC2)n3C)c1C(=O)NCc1cc(CO)no1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CNc1cc2oc(-c3cncc(CNC(=O)NCc4ccc(OC)c(OC)c4)c3)nc2cn1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CNc1ccc(OCCNC(=O)Cc2cc(-c3cc4ccccc4c(=O)[nH]3)on2)c(C#N)n1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 CNC(=O)c1ccn(C(=O)Cc2nn(C)c3ccc(NC(=O)Nc4ccc(O)cc4)cc23)c1
C(=O)(Nc1n[nH]cc1)OCc1ccc(cc1)c1[nH]c2c(n(c(=O)n(c2=O)CCC)CCC)c1 O=C(Nc1c[nH]nc1O)N(CCn1ncc(CCCc2ccccc2)n1)c1cccc(O)c1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C Cc1[nH]c(-c2noc(-c3cc(N(C)C)ccc3OCCO)n2)cc1COc1ccc2[n+](c1)CCN=C2
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCCOCCN(CCC)C(=O)c1nn(-c2nc(=O)c3ccccc3[nH]2)c(-c2cccc(OC)c2)[nH+]1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C C[NH2+]Cc1ccc(OC)nc1C(=O)OCCC(=O)c1ccc(C)c(-n2nc(C)c3nc(C)cnc32)c1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCC(C)[NH+](CCOC)Cc1nc2cc(CNC(=O)C=Cc3nnc(-c4ccn(C)c4)o3)ccc2o1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCOc1ccccc1NC(=O)c1cc(OCc2cc[nH+]c(-n3c(C)nnc3C)c2)nc(COC)n1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCCCNC(=O)c1cc(OCC(=O)n2c(-c3nnc(C[NH+](C)C)o3)cc3ccccc32)ncc1C
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C COCC[NH+](Cc1n[nH]c(-c2ccc(Oc3ccc(OC)nc3)nc2)n1)C(C)c1ccc(OC)cc1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C C=C(C)c1nc(CCn2c(C=Cc3ccc(C)o3)nnc2NC(=O)C[NH+](CC)Cc2ccco2)co1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCC(C)[NH2+]CC(=O)c1ccc(-c2nc3n(C(=O)COc4ccc(C)cc4OC)nc(C)n3n2)cc1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C COC(C)c1nn(C)c(=O)n1-c1ccc(C[NH2+]Cc2cc(C(=O)N(C)c3ccccc3)c(C)o2)cn1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCOCCOc1nn(C)[nH+]c1C(=Nc1ccccn1)NC(C)Cc1cc2ccoc2cc1OCC
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C C=N[NH+](CC)CC(=O)c1ccc(-c2cc(Nc3nc4ccc(C(C)C(=O)OC)cc4o3)n(C)n2)cc1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCC(C)OCCn1c(Cn2n[nH+]cc2C)nc2cc(NC(=O)COc3cccc(OC)c3)ccc21
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCCC[NH+](CCNC(=O)c1ccc(O)cc1)Cc1noc(C=C(c2ccoc2C)n2cccn2)n1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C C[NH2+]CC(c1ccco1)n1ccc(C)nc1=NC(=O)c1cnn(-c2ccc(OCCOC)cc2)c1C
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C COc1cc(OC(C)c2nnc(-c3ccc(C)cc3C)n2CCC(C)O)cc2c(=O)n(C)[nH+]cc12
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C C[NH2+]Cc1c(C)cc(C)nc1Oc1ccc(-c2c(CCCn3cnn(CCO)c3=O)noc2C)cc1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C C[NH2+]Cc1cc(N(Cc2ccc(C)cc2)C(=O)c2ccc(-c3nnc(C(C)CCOC)o3)o2)n(C)n1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C C=C1OCC=C1Cn1[nH+]c(NC(COc2ccccc2OC)Cc2ccc(OC)cc2)n2ncnc12
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CC(COCc1ccc(CNC(=O)Nc2ccc(Oc3ncc4ccncc4n3)cc2)o1)[NH+](C)C
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C COc1ccc(C)c(OC(=O)C[NH2+]c2ccc(-n3c(C=CN(C)C)nnc3-c3ccno3)cc2)c1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C COCC(=O)N(C[NH+](Cc1cocc1C)Cc1cn(C)c2ncccc12)C(=O)NCc1ccncc1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CC[NH+](C)CC=CC(OC(=O)c1ccc(-n2nnc3cc(C)[nH]c(=O)c32)nc1)c1ccc(C2CC2)o1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCOc1nc(C[NH+](C)C(C)CCC=CCNC(=O)n2c(-c3ccc(C)o3)nc3ccccc32)no1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CC[NH+](Cc1cnc(-c2c(OC)cnc(N(C)C)c2C)c(O)c1)Cc1nnc(-c2ccc(O)cc2)o1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C COc1cc(C[NH2+]CCCCc2nc(-c3cnn(C)c3)no2)cc(OC)c1Oc1ccc(C)nc1C
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCN(CCOC)c1[nH+]c(-c2ccccc2)ccc1CNc1nc(COC(=O)c2ccncc2)no1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C C=CC[NH+](Cc1ncco1)Cc1nc(-c2ccc(Oc3ccc(NC(=O)C(C)CC)cc3)nc2)no1
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C CCOc1cc(C)cc(N(Cc2c[nH+]cc(O)c2)c2ccc(C(=O)Nc3cnn(C)c3)nc2)c1OC
c1(nc(nc(c1)NC(=O)COc1c(cc(cc1)C[NH+](C)C)OC)c1ccc(o1)C)n1nc(cc1C)C Cn1cc(C=Nc2occ(C=CC(=O)Nc3ccc4nc(C5CCOC5)oc4c3)c2C[NH+](C)C)cn1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F COc1ccc(F)cc1-n1cnc(SC(C)C(O)=CF)c(C=Nc2ccc3cnc(F)cc3n2)c1=O
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F Cc1nc(C(F)(F)F)c(CCN(Cc2cc(O)ccn2)C(=O)c2ccnc(Oc3cccnc3)c2)s1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CCc1ccc(-c2cc(S(=O)(=O)Nc3ccc(F)c(-n4nnnc4C(F)F)c3)cc(C=O)c2C)cc1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F COc1cccc(F)c1N=C(Oc1ccncc1O)SCc1nc(C)nn1Cc1cc(F)cc(F)c1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CCc1nocc1C=CCc1nc(SCCOc2cccc(C(F)(F)F)n2)nc2cc(C)[nH]c(=O)c12
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CCCOc1ncc(C(F)F)cc1S(=O)(=O)Nc1cc(F)cc(-n2ncc3cc4c(nc32)CCC4)c1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F N#CCn1cc(F)cc(OCCc2ncc(CSc3ccc4ccc(NCC(F)F)cc4n3)o2)c1=O
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F C=Cc1nc(C)cc(Nc2cc(F)c(OC3(F)OCc4cc5nc(N(C)C)sc5cc4O3)c(F)c2)n1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F Cn1cc(-c2ccc(SCCOc3ccc(C(=O)Nc4ccncc4)nc3)cc2OC(F)(F)F)cn1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CCOCc1cc(-c2nnc(Sc3ccc(C(=O)NN=Cc4ccc(F)c(F)c4)cc3)o2)cnc1F
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F Cc1ccc2cc(C(=O)Nc3nnc(CC(C)C(F)F)s3)cc(C(=O)OCc3nccc(F)n3)c2c1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F COCC=CN(Cc1sc(=NC(=O)c2cccc(F)c2F)[nH]c1C)c1cc(F)ccc1-c1nnco1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F COc1nc(Oc2ccc[nH]c2=O)cc(Cn2c(SCc3cc(C)cc(C)c3)nnc2C(F)F)c1F
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F COc1cc(C(F)F)cc(F)c1OCC(=O)N=c1[nH]c(-c2ccc(C)cc2)c(C=Nn2ccnc2)s1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F COC(=O)C=Cc1ccc(CSCc2nc(Nc3ccc(F)nc3)n(-c3ccc(F)cc3C)n2)o1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F Cc1cnc(N=c2sc3cc(OCF)c(F)cc3n2NC(=O)c2ccc(OCC#N)c(C)c2)c(F)c1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CN(C(=O)C(=Cc1ccncc1)N(CCOc1ccncc1O)c1nc2ccccc2s1)C(F)(F)F
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CCc1nnc(N(CCN(CC)S(=O)(=O)Nc2ccc(F)c(F)c2F)c2cccc3ccccc23)o1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F Cc1ncn(-c2c(NC(=O)C(=Cc3ccc(C(F)F)o3)SCC=Cc3ccc(C)o3)ccnc2F)n1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CCc1cc(OC(F)(F)F)c(COc2cc(C(=O)Nc3cnn(-c4nc(C)cs4)c3)ccn2)cc1C
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F C=C(OF)c1cc(F)c(NC(=O)Cc2csc(C(=O)N(C)c3ccc(-n4cccn4)cc3)n2)cc1F
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F N#Cc1ccc(CN(CC2COCCO2)c2cc(F)cc(-c3ncc(-c4c[nH]c(C(F)F)n4)s3)c2)o1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F Cc1ccc(COc2ccc(OCC(=O)N=c3[nH]c(-c4cc(C(F)F)n(C)c4C)ns3)c(F)c2)cn1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F C=NC(=CF)c1ncn(Cc2cc(C(=O)c3c(C)c(C(=O)Oc4ccc(F)c(F)c4)cn3C)cs2)n1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CC=CC(=O)N(CC(C)c1noc(-c2cc(NC(=O)C(F)(F)F)cs2)n1)c1nccc2ccccc12
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CC(OC(=O)c1ccnc(F)c1-c1ccc(-n2ncnc2SC(F)F)cc1)C(=O)Nc1ccccc1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F Cc1c2c(nn1-c1nnc(SCC(=O)c3cc(F)c(Oc4ccccc4)c(F)c3)[nH]1)CCCC2=O
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F CN(C)C(=O)c1cccc(-n2nnc3cc(NC(=O)CSc4ccc(OC(F)(F)F)cc4)ccc32)c1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F Cc1ccc(N(C)C(=O)COc2ccc(-c3nnc(CSc4ncc[nH]4)o3)c(CC(F)(F)F)c2)cc1
c1cc(N(C(=O)C)CC)c2c(c1OC)nc(s2)NC(=O)c1cn(nc1)Cc1cccc(c1)C(F)(F)F C=C(F)C(=CC)Cn1cnc(C(OC(=O)c2ccc(F)cc2F)C(=O)N=c2[nH]c3ccccc3s2)n1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 N#CCc1ccc(C(=O)N(CCC(=O)N2CCCc3ccccc32)c2ccc(NC(=O)[O-])cc2)cc1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 N#Cc1ccc2ccc(CN(CCC(=O)N3CCCCC3)C(=O)Nc3cccc(C(=O)[O-])c3)cc2c1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 Cc1cc(NC(=O)c2cc(C)c3ccccc3c2)ccc1C(=O)N=C(N1CCC(C)C1)N(C)C(=O)[O-]
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 Cc1ccc(C=Cc2nc(C3CN(C(=O)N4c5ccc(CC(=O)[O-])cc5CC4C)CCO3)c[nH]2)cc1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CCC1Cc2ccc(C)cc2C(COc2ccc(C(=O)N3CCc4nc([O-])[nH]c(=O)c4C3)c(C)n2)C1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CC(=CC(=O)N1CC2C([O-])=NN=C(O)C2C1)c1ccc(-c2cc3ccccc3n(C(C)C)c2=O)cc1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 C=CCN1C(=O)c2ccc(NC(=O)C(C#N)=Cc3ccc(C#N)cc3)c3cc(C)c([O-])c(c23)C1=O
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CN(C=NN=Cc1ccc(C(=O)Nc2cccc(C(=O)[O-])c2)cc1)C(=O)c1ccc2c(c1)CCC2
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CC=CC=CC(=O)c1ccc2c(NCN3C(=O)C(=C[O-])N(c4ccc(C#N)cc4)C3=O)cccc2c1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 Cc1ccccc1Cc1cccc(C=C2C(=O)NC(=O)N(c3cc([O-])c(N(C)C)c(C#N)c3)C2=O)c1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 N#CC(=Cc1cccc(C(=O)[O-])c1)C(=O)Nc1ccc(N=C(c2ccccc2)N2CCOCC2)cc1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 Cc1ccc(C2c3ccccc3CN2C(=O)N(C)c2cc(C#N)ccc2NC(=O)CCC(=O)[O-])cc1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CC1CCCC(NC(=O)c2ccc(-n3c([O-])c(C#N)c(=O)n(-c4ccc(C(C)C)cc4)c3=O)cc2)C1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 O=C([O-])c1ccc2c(ccn2CC(=O)N2CCCCC2C(=O)Nc2ccccc2N2CCCCC2)c1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CCC1C=CC2CN(C=NC(=O)c3ccc([O-])c4cccc(NC(=O)c5cccn(C)c5=O)c34)CC12
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 C=CC(=CC)C(=O)C=Cc1c(CN2CCOCC2)c(=O)[nH]c2nc([O-])c(C#N)c(-c3ccccc3)c12
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 C=CCN(C(=O)c1ccnc(C(=O)[O-])c1)c1ccc(C(C)(C)C)c(C(=O)N=CNc2ccccc2)c1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 O=C([O-])c1cccc(NC(=O)c2ccc(CC(=O)N(c3cnn(C4CCCC4)c3)C3CCC3)cc2)c1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CC(C)(C)CCC1CN(c2nccc3c(C=C(CCC(=O)[O-])c4ccccc4)n[nH]c(=O)c23)CCO1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 Cc1c(C(=O)[O-])c(C2CCCN2C(=O)CC=CC2CCC2)nc2[nH]c(=O)n(C=Cc3ccccc3)c12
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 Cc1cccc(NC(=O)c2cccc(C#CC(=O)N(CCC#N)c3ccc(C)c(C(=O)[O-])c3)c2)c1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 C=CCNC(=O)C1CCC(C#N)CN1C(=O)C=Cc1ccc(-c2ccc(-c3conc3[O-])cc2)cc1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 N#Cc1ccc(CC2CCCN2C(=O)NCc2cc(-c3ccc(C#N)cc3)ccc2OC(=O)[O-])cc1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 Cc1cnc(N2CC3CCCc4cccc2c43)c(C(=O)Nc2ccccc2CN(C)C(=O)C(=O)[O-])c1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CC(=CC1OCCC12CCC2)Cn1ccc(N(CCC(=O)[O-])C(=O)Nc2cccc3ccccc23)n1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CC(C)(C)c1ccc(NC(=O)C(C#CC(=O)[O-])=Cc2ccc(C(=O)Cc3ccn(C#N)n3)cc2)cc1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 COc1cc(C=Cc2ccc3c(c2)CCCC3)cc(C=C(C(=O)[O-])c2nc3n(n2)C(C)CC(=O)N3)c1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 COc1c([O-])cccc1C(=O)N1CC2Nc3cc(C(=O)N4CCCc5cc(C)ccc54)ccc3N2C1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 CN1CCOC(CN(C(=O)c2cccc(NC(=O)c3ccnc([O-])c3)c2)C2CCc3ccccc32)C1
c12n(c(=O)n(c(=O)c1nc([nH]2)c1ccc(/C=C/C(=O)[O-])cc1)CC1CCCCC1)CC1CCCCC1 Cn1nc(Cc2ccc3c(c2)CCC(C(C)(C)C)C3)c2c1NC(=O)C(CC(=O)[O-])N2Cc1ccco1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CNc1ccc2c(NC(=O)C(=O)NC(C)(CCO)CCc3ccc(Cc4ccc(N=c5[nH]ccn5C)cc4)cc3)cnnc2n1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CCN(C)C(=O)C(O)Cc1ccc(Nc2nc(N)c3c(C)cc4cc(C(=O)NCCn5cnnc5C)ccc4c3n2)cc1C
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CCC(=N)NCc1ccc(-n2nc(C)c(NC(=O)CNC(=O)CNC(=O)c3c4ccccc4cc4[nH]nc(C)c34)c2C)c(C)c1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC C=CC(=C)NC(c1cc(NC(=O)c2cc(CNC(=O)c3ccc(Cc4ncnn4C)cc3)cn2C)ccn1)c1ccc[nH]c1=O
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1c(NC(=O)C(=O)NN=c2[nH]c3ccccc3n2C)cccc1C(=O)NN=Cc1cc(C)n(CCNc2ccccc2)c1C
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1cc(C(=O)N(C)CC2CC(C)C(C)N2)cc2c(Oc3cc(NCCCO)nc(Nc4nc[nH]n4)n3)cc3ccccc3c12
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CCc1ccc(Nc2cc(CNc3cc(NC(=O)CN4CC(C)n5c(n[nH]c5=O)C4=O)ccc3C)n[nH]2)c2cc(C)c(C)cc12
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1c(C(=O)NNc2cc(C#N)ccc2-n2ccnc2)c(C(=O)OC(C)c2ccnc(NCCN)c2)c(C)n1-c1ccccc1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1ccc(C#N)cc1NC(=O)Cc1ccc2c(c1)cc(C)n2C(=O)c1ccc(C(=O)NN=Cc2cc[nH]c2NCCN)cn1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CCN1Cc2c([nH]c3c4c(nn23)C(=O)NC(C(C(=O)Oc2cccc(C)c2)=C(C)Nc2c3c(C)c(C)[nH]c3nn2C)C4)CC1C
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1ncnc2c1c(N)nc(=O)n2Cc1ccccc1-c1cc(-c2cccc(CCC(=O)NC(CC#N)CC(C)O)c2)nn1C
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC C#CCN(CCc1cc(C)n[nH]1)C(=O)c1cc2cccnc2cc1C(=O)Nc1nc(C)c(C)cc1C(=O)NNc1ccncc1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1ccc(-c2c(C(=O)N3CCc4cc(C)ccc43)nc3ncc(=Cc4cnc(NCCC(CO)NC(=O)CN)nc4)n23)cc1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1cnc2ncc3ccc(Oc4ccc(C(=O)NCc5cc(C#N)cc(NC(C(=O)NN=CN)C(C)C)c5)cn4)cc3c2c1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC C=c1[nH]c2c(C(CO)Nc3c(CN(C)C=NC=CC)cc(OCCN4CCn5c(C)nnc5C4)cc3C(N)=O)cccc2c1=C
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CCC1=Nc2c([nH]c(=O)c3cnn(CC(O)CNN)c23)C1=Cc1ccc(Oc2ccc(-c3nn(C)c(C)c3CC)cc2)cc1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1cc(-c2ncc(NCCc3ccc(C(=O)Nc4ccc(C(C)n5c(C)nc(C(C)C#N)cc5=O)cc4)cc3)c(=O)[nH]2)[nH]n1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CNc1cccc(CNC(C)=C(C(=O)N(CC(=O)N=c2[nH]cc[nH]2)Cc2cc(C(C)=O)[nH]n2)C(C)=CN=Cc2ccccc2)c1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC COc1ccc(C=CCC(=O)NN=Cc2ccccc2-c2nc(NCc3cc(=O)[nH]c(N)n3)n(-c3ccc(C)cc3)n2)cc1C
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CNCc1cc(CNC(=O)c2ncc(N(CC(=O)N(CCC#N)c3cc[nH]c(=O)c3)c3ccncc3)cc2C)ccc1C=CN
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1[nH]c(C(=O)NCCN(Cc2ccccn2)Cc2nccn2C)c(C)c1C(=O)c1ccc(NC(=O)Nc2cccnc2)cc1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CCCc1ccc(C(CN(C)c2ncccc2-n2c(N)n[nH]c2=Nc2cccc(C(N)=O)c2)Oc2cccnc2OCC)cc1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1nc2nc3n(C4CCCC4)c(Nc4ccc(C(CCO)CNNCN)[nH]4)c(C)n3c(=O)c2cc1C(=O)Cc1ccccc1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1ccc(C=Cc2nc(C(=O)C(c3cccnc3)n3cc(C(=O)NCc4ccnc(N)c4)n(C4CC4)c3=O)n[nH]2)cc1C
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CNCc1ccc(C(=O)Nc2ccc(NC(=O)Nc3nc(OC)c4ccccc4n3)cc2)c(N(CCC#N)Cc2ccc[nH]2)n1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC Cc1ccc(C)c(NCc2nc(C(=O)NCc3c[nH]c4ccc(C(C)C#N)cc34)c(CCCn3ncc(C(N)=O)c3C)o2)c1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CNC(=O)C(=O)Nc1cccc(C(Nc2ccc3ccn(C)c3c2)c2cccc(C(=O)NN=Cc3c(C)nn(C)c3C)c2)c1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CCCCCCc1nc(C=CC(C)Oc2cc(C)cc(C)c2)n(-c2nc3c(-c4ncc[nH]4)c(N)[nH]c3c3c2C(=O)NC3=O)n1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CN(CC#N)c1ccc(NC(=O)CNc2nc3nc(OC(C)(c4ccccc4Oc4ccc(N)cc4)N(C)C)ccc3[nH]2)cc1
N([C@@H]1[C@H]([C@H]([C@H](n2c3nc(nc(c3nc2)NCC(c2ccccc2)c2ccccc2)NCCc2cn(cn2)C)C1)O)O)C(=O)CC CCN(CCNc1cccc(-n2cncn2)c1)C(=O)c1ccccc1N(CC)C(=O)CNc1ccc2c(N)ccc(C)c2n1
